SCHEMBL7307254

SCHEMBL7307254

CC(C)(C)OC(=O)C[C@H](NC(=O)CCCc1ccc(C(N)=S)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.49
MMP3 P08254 1/20 0.49
MMP9 P14780 1/20 0.49
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
MAPT P10636 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
REN P00797 1/20 0.42
ACE P12821 1/20 0.42
KLK5 Q9Y337 1/20 0.42
POLB P06746 1/20 0.42
CAPN1 P07384 1/20 0.42
CTSG P08311 1/20 0.41
CMA1 P23946 1/20 0.41
HDAC1 Q13547 4/20 0.41
HDAC6 Q9UBN7 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9218199 0.88 MMP1 (0.49) MMP1MMP3MMP9MAPTTDP1
SCHEMBL7307169 0.88 CCKBR (0.44) MMP1MMP3MMP9MAPTTDP1
SCHEMBL7302254 0.87 TDP1 (0.46) MMP1MMP3MMP9MAPTTDP1
SCHEMBL9223666 0.85 REN (0.49) MAPTTDP1RENKLK5
SCHEMBL8438729 0.82 MEN1 (0.47) MMP1MMP3MMP9MAPTTDP1
SCHEMBL9215215 0.82 ITGB3 (0.52) MMP1MMP3MMP9ITGB3ITGA2B
SCHEMBL9339365 0.81 MAPT (0.45) ITGB3ITGA2BMAPTTDP1REN
Iodide SCHEMBL9215204 0.81 ITGB3 (0.51) MMP1MMP3MMP9ITGB3ITGA2B
SCHEMBL9218412 0.80 ST14 (0.47) MMP1MMP3MMP9ITGB3ITGA2B
Iodide SCHEMBL9218396 0.79 ST14 (0.47) MMP1MMP3MMP9ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed