SCHEMBL7308041

SCHEMBL7308041

O=C(O)CC1(Sc2ccc(Oc3ccc(F)cc3)cc2)CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KDM1A O60341 2/20 0.43
OPRK1 P41145 2/20 0.42
HTR1A P08908 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
HTR2C P28335 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CYP2C19 P33261 1/20 0.41
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
OPRD1 P41143 1/20 0.39
SCN5A Q14524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308120 0.94 OPRK1 (0.47) MEN1KMT2ANPSR1KDM1AOPRK1
SCHEMBL7301926 0.91 HDAC1 (0.43) RORCMEN1KMT2ANPSR1KDM1A
SCHEMBL7311907 0.88 P2RX7 (0.41) RORCMEN1KMT2ANPSR1KDM1A
SCHEMBL7303615 0.87 SCN5A (0.49) MEN1KMT2ANPSR1KDM1AOPRK1
SCHEMBL7308906 0.78 MMP9 (0.51) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL471541 0.76 RORC (0.49) RORCMEN1KMT2ANPSR1KDM1A
SCHEMBL7302125 0.75 ALDH1A1 (0.39) MEN1KMT2ASLC6A3SCN9A
SCHEMBL7312678 0.75 MMP1 (0.43)
SCHEMBL7303726 0.73 ALDH1A1 (0.44) MEN1KMT2A
SCHEMBL8696969 0.73 RORC (0.58) RORCMEN1KMT2ANPSR1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed