SCHEMBL7313718

SCHEMBL7313718

CC(C)(C)OC(=O)NC(=N)N1CCN(CCN2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.31
MAPK1 P28482 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
CD274 Q9NZQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310460 0.95 SIGMAR1 (0.34) SIGMAR1MAPK1L3MBTL1
SCHEMBL7313917 0.95 SIGMAR1 (0.34) SIGMAR1MAPK1L3MBTL1
SCHEMBL7314189 0.89 GPR119 (0.33)
SCHEMBL7313885 0.87 GPR119 (0.38) MAPK1L3MBTL1
SCHEMBL7307684 0.86 GPR119 (0.39) MAPK1L3MBTL1
SCHEMBL7236582 0.86 CHRM2 (0.38)
SCHEMBL7308728 0.82 SIGMAR1 (0.34) SIGMAR1CD274
SCHEMBL7303526 0.82 SIGMAR1 (0.33) SIGMAR1CD274
SCHEMBL7235475 0.82 USP30 (0.32)
SCHEMBL7315937 0.81 ITGB3 (0.35) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed