SCHEMBL7314189

SCHEMBL7314189

CC(C)(C)OC(=O)NC(=N)N1CCC(CCN2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 11/20 0.33
RORC P51449 6/20 0.32
SCN9A Q15858 1/20 0.31
FAAH O00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313885 0.95 GPR119 (0.38) GPR119SCN9AFAAH
SCHEMBL7307684 0.94 GPR119 (0.39) GPR119RORCFAAH
SCHEMBL7313718 0.89 SIGMAR1 (0.31)
SCHEMBL7313917 0.87 SIGMAR1 (0.34)
SCHEMBL7310460 0.87 SIGMAR1 (0.34)
SCHEMBL7235475 0.85 USP30 (0.32) GPR119
SCHEMBL7317037 0.81 DRD2 (0.33) RORC
SCHEMBL7316461 0.80 DRD2 (0.34) RORCFAAH
SCHEMBL7316825 0.80 ITGB3 (0.34) RORC
SCHEMBL7310067 0.80 DRD2 (0.33) FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed