Isoformonentin

Isoformonentin

SCHEMBL73338

COc1ccc2c(=O)c(-c3ccc(O)cc3)coc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 1.00
MAOA P21397 7/20 0.85
MAOB P27338 7/20 0.85
MAPT P10636 4/20 0.85
KDM4E B2RXH2 4/20 0.85
ALDH1A1 P00352 4/20 0.85
CYP3A4 P08684 4/20 0.85
HPGD P15428 4/20 0.85
TP53 P04637 3/20 0.85
SMN1; SMN2 Q16637 3/20 0.85
HSD17B10 Q99714 3/20 0.85
HDAC6 Q9UBN7 3/20 0.85
MEN1 O00255 2/20 0.85
KMT2A Q03164 2/20 0.85
CYP2D6 P10635 2/20 0.85
CYP2C9 P11712 2/20 0.85
CYP2C19 P33261 2/20 0.85
BCL2 P10415 1/20 0.85
IL2 P60568 1/20 0.85
CYP1B1 Q16678 1/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isoformonentin SCHEMBL30105310 1.00 XDH (1.00) XDHMAOAMAOBMAPTKDM4E
Formononetin SCHEMBL8416577 0.93 KDM4E (0.97) XDHMAOAMAOBMAPTKDM4E
Formononetin SCHEMBL62915 0.92 KDM4E (1.00) XDHMAOAMAOBMAPTKDM4E
Formononetin SCHEMBL29361145 0.92 KDM4E (1.00) XDHMAOAMAOBMAPTKDM4E
Formononetin SCHEMBL15271536 0.92 KDM4E (1.00) XDHMAOAMAOBMAPTKDM4E
SCHEMBL571576 0.92 XDH (0.84) XDHMAOAMAOBMAPTKDM4E
Formononetin SCHEMBL6638953 0.91 KDM4E (0.97) XDHMAOAMAOBMAPTKDM4E
SCHEMBL5814089 0.88 XDH (0.78) XDHMAOAMAOBMAPTKDM4E
SCHEMBL32659701 0.87 XDH (0.77) XDHMAOAMAOBMAPTKDM4E
SCHEMBL13774686 0.86 XDH (0.76) XDHMAOAMAOBMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 126 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160068542-A1 Enhanced Osteogenic Activity of Daidzein Analogs on Human Mesenchymal Stem Cells THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF AGRICULTURE 2016-03-10 US claimed
EP-2981530-A2 ENHANCED OSTEOGENIC ACTIVITY OF DAIDZEIN ANALOGS ON HUMAN MESENCHYMAL STEM CELLS The Administrators of the Tulane Educational Fund (US) 2016-02-10 EP claimed
US-20150148409-A1 NOVEL DAIDZEIN ANALOGS AS TREATMENT FOR CANCER XAVIER UNIVERSITY OF LOUISIANA 2015-05-28 US claimed
US-8962679-B2 Daidzein analogs as treatment for cancer THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2015-02-24 US claimed
WO-2014165723-A2 ENHANCED OSTEOGENIC ACTIVITY OF DAIDZEIN ANALOGS ON HUMAN MESENCHYMAL STEM CELLS THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2014-10-09 WO claimed
US-20130184475-A1 NOVEL DAIDZEIN ANALOGS AS TREATMENT FOR CANCER THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2013-07-18 US claimed
WO-2012006563-A2 NOVEL DAIDZEIN ANALOGS AS TREATMENT FOR CANCER THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2012-01-12 WO claimed
EP-2278882-A2 COMPOSITIONS AND METHODS TO CONTROL OOMYCETE FUNGAL PATHOGENS Dow AgroSciences LLC (US) 2011-02-02 EP claimed
WO-2009146079-A2 COMPOSITIONS AND METHODS TO CONTROL OOMYCETE FUNGAL PATHOGENS DOW AGROSCIENCES LLC (US) 2009-12-03 WO claimed
US-20090246293-A1 COMPOSITIONS AND METHODS TO CONTROL OOMYCETE FUNGAL PATHOGENS DOW AGROSCIENCES LLC (US) 2009-10-01 US claimed
CN-122097338-A Application of formononetin in preparation of medicines for preventing and treating depression 2026-05-29 CN disclosed
US-12507703-B2 Methods, devices and compositions for preserving human milk THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2025-12-30 US disclosed
US-20250169516-A1 METHODS, DEVICES AND COMPOSITIONS FOR PRESERVING HUMAN MILK THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2025-05-29 US disclosed
US-12239142-B2 Methods, devices and compositions for preserving human milk THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2025-03-04 US disclosed
US-20240268402-A1 Methods, Devices and Compositions for Preserving Human Milk THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2024-08-15 US disclosed
WO-2004002470-A1 COMPOUNDS USEFUL FOR THE INHIBITION OF ALDH THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 2004-01-08 WO disclosed
WO-2003006987-A9 METHODS AND COMPOSITIONS FOR DETERMINING ENZYMATIC ACTIVITY AND SPECIFICITY OF METHYLTRANSFERASES SALK INST FOR BIOLOGICAL STUDI (US) 2003-04-24 WO disclosed
WO-2003006987-A1 METHODS AND COMPOSITIONS FOR DETERMINING ENZYMATIC ACTIVITY AND SPECIFICITY OF METHYLTRANSFERASES THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2003-01-23 WO disclosed
EP-1183376-A1 ISOFLAVONOID METHYLATION ENZYME The Samuel Roberts Noble Foundation, Inc. (US) 2002-03-06 EP disclosed
WO-2000071736-A1 ISOFLAVONOID METHYLATION ENZYME THE SAMUEL ROBERTS NOBLE FOUNDATION, INC. (US) 2000-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12507703-B2 Methods, devices and compositions for preserving human milk LPL, CEL, LPO XDH 171/4885MAOA 471/4885MAOB 293/4885
US-20160068542-A1 Enhanced Osteogenic Activity of Daidzein Analogs on Human Mesenchymal Stem Cells HPGDS, CXCL12, ALPG XDH 1126/4885MAOA 2979/4885MAOB 2571/4885
US-20090246293-A1 COMPOSITIONS AND METHODS TO CONTROL OOMYCETE FUNGAL PATHOGENS ERG28, DPM1, CYP51A1 XDH 323/4885MAOA 266/4885MAOB 295/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.