SCHEMBL734966

SCHEMBL734966

[CH2]COC(=O)Nc1cccc2ccccc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.72
HPGD P15428 1/20 0.72
KDM4E B2RXH2 5/20 0.57
GAA P10253 1/20 0.57
LMNA P02545 2/20 0.56
MAPT P10636 3/20 0.54
KMT2A Q03164 3/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
NPC1 O15118 4/20 0.53
RAB9A P51151 3/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2C19 P33261 2/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
GSK3B P49841 1/20 0.51
EPHX1 P07099 1/20 0.50
MEN1 O00255 1/20 0.50
POLB P06746 1/20 0.49
TSHR P16473 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL283472 0.84 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL9271743 0.83 ALDH1A1 (0.67) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL10401087 0.83 ALDH1A1 (0.70) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL2094345 0.81 ALDH1A1 (0.64) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL10959203 0.81 HPGD (0.78) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL9523920 0.81 ALDH1A1 (0.68) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL10959557 0.80 ALDH1A1 (0.71) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL283066 0.80 ALDH1A1 (0.71) ALDH1A1HPGDKDM4EGAALMNA
SCHEMBL9813594 0.79 ALDH1A1 (0.74) ALDH1A1HPGDKDM4EGAALMNA
Acrylic Acid SCHEMBL17822133 0.79 ALDH1A1 (0.82) ALDH1A1HPGDKDM4EGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117264004-A Compound and nucleic acid synthesis method 深圳华大生命科学研究院 2023-12-22 CN claimed
CN-110678447-B Modified nucleic acid monomer compounds and oligonucleotide analogues 卫材R&D管理有限公司 2023-12-12 CN claimed
EP-3643706-B1 MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES EISAI R&D MAN CO LTD (JP) 2023-11-15 EP claimed
US-9714560-B2 Protected scale inhibitors and methods relating thereto HALLIBURTON ENERGY SERVICES, INC. (US) 2017-07-25 US claimed
US-20020147331-A1 Methods for synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. 2002-10-10 US claimed
WO-2002062811-A2 IMPROVED METHODS FOR SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2002-08-15 WO claimed
CN-117264004-A Compound and nucleic acid synthesis method 深圳华大生命科学研究院 2023-12-22 CN disclosed
CN-110678447-B Modified nucleic acid monomer compounds and oligonucleotide analogues 卫材R&D管理有限公司 2023-12-12 CN disclosed
EP-3643706-B1 MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES EISAI R&D MAN CO LTD (JP) 2023-11-15 EP disclosed
US-11208429-B2 Modified nucleic acid monomer compound and oligonucleic acid analog EISAI R&D MANAGEMENT CO., LTD. (JP) 2021-12-28 US disclosed
US-10874740-B2 5-ALA derivatives and use thereof UNIVERSITE DE GENEVE (CH) 2020-12-29 US disclosed
EP-3643706-A9 MODIFIED NUCLEIC ACID MONOMER COMPOUND AND OLIGONUCLEIC ACID ANALOG Eisai R&D Management Co., Ltd. (JP) 2020-09-23 EP disclosed
US-20200216488-A1 MODIFIED NUCLEIC ACID MONOMER COMPOUND AND OLIGONUCLEIC ACID ANALOG EISAI R&D MANAGEMENT CO., LTD. (JP) 2020-07-09 US disclosed
EP-2915815-A1 NEW MODIFIED NUCLEIC ACID Takeda Pharmaceutical Company Limited (JP) 2015-09-09 EP disclosed
WO-2014200757-A1 PROTECTED SCALE INHIBITORS AND METHODS RELATING THERETO HALLIBURTON ENERGY SERVICES, INC. (US) 2014-12-18 WO disclosed
US-20140367101-A1 Protected Scale Inhibitors and Methods Relating Thereto HALLIBURTON ENERGY SERVICES, INC. 2014-12-18 US disclosed
US-8138330-B2 Solid phase synthesis via deblocking immobilized nucleoside, then coupling acyl protected nucleoside phosphoramidite SIGMA-ALDRICH CO. LLC (US) 2012-03-20 US disclosed
US-20080064867-A1 PROCESS FOR THE SYNTHESIS OF OLIGONUCLEOTIDES SIGMA ALDRICH COMPANY (US) 2008-03-13 US disclosed
US-20020147331-A1 Methods for synthesis of oligonucleotides ISIS PHARMACEUTICALS, INC. 2002-10-10 US disclosed
WO-2002062811-A2 IMPROVED METHODS FOR SYNTHESIS OF OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 2002-08-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200216488-A1 MODIFIED NUCLEIC ACID MONOMER COMPOUND AND OLIGONUCLEIC ACID ANALOG POLRMT, DERA, PCNA ALDH1A1 2175/4885HPGD 1535/4885KDM4E 3391/4885
US-20080064867-A1 PROCESS FOR THE SYNTHESIS OF OLIGONUCLEOTIDES RNGTT, DUT, ADAR ALDH1A1 2127/4885HPGD 4031/4885KDM4E 1717/4885
US-11208429-B2 Modified nucleic acid monomer compound and oligonucleic acid analog POLRMT, DERA, PCNA ALDH1A1 2175/4885HPGD 1535/4885KDM4E 3391/4885
US-10874740-B2 5-ALA derivatives and use thereof ALAD, ANXA5, AAAS ALDH1A1 76/4885HPGD 249/4885KDM4E 1819/4885
US-20020147331-A1 Methods for synthesis of oligonucleotides RNGTT, TYMP, PNP ALDH1A1 4843/4885HPGD 3858/4885KDM4E 4628/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.