SCHEMBL7357115

SCHEMBL7357115

CC(C)(C)NS(=O)(=O)Nc1ccc(-c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
UQCRB P14927 2/20 0.46
ALDH1A1 P00352 4/20 0.45
NR3C2 P08235 2/20 0.45
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PGR P06401 1/20 0.43
KEAP1 Q14145 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
PLAU P00749 1/20 0.41
KIF11 P52732 4/20 0.41
USP30 Q70CQ3 1/20 0.41
MCL1 Q07820 1/20 0.40
MEN1 O00255 1/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491328 0.89 KEAP1 (0.54) ALDH1A1NR3C2MAPTSMN1; SMN2KEAP1
SCHEMBL13141234 0.78 ALDH1A1 (0.51) UQCRBALDH1A1NR3C2MAPTSMN1; SMN2
SCHEMBL7547560 0.77 KIF11 (0.47) KIF11
SCHEMBL7545504 0.77 ACLY (0.48) KIF11
SCHEMBL7338377 0.75 LMNA (0.45) ALDH1A1MAPTSMN1; SMN2PGRCYP3A4
SCHEMBL873846 0.75 KEAP1 (0.75) UQCRBALDH1A1NR3C2SMN1; SMN2PGR
SCHEMBL27802067 0.74 ALDH1A1 (0.56) UQCRBALDH1A1MAPTSMN1; SMN2CYP3A4
SCHEMBL8530361 0.74 CA1 (0.56) ALDH1A1MAPTSMN1; SMN2PGRCYP3A4
SCHEMBL11676103 0.74 MAPT (0.55) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL23141160 0.71 KEAP1 (0.61) ALDH1A1NR3C2MAPTPGRKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216231-A2 INHIBITORS OF FACTOR Xa Millennium Pharmaceuticals, Inc. (US) 2002-06-26 EP disclosed
WO-2001019798-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC. (US) 2001-03-22 WO disclosed
EP-0991638-A1 NOVEL GUANIDINE MIMICS AS FACTOR Xa INHIBITORS Du Pont Pharmaceuticals Company (US) 2000-04-12 EP disclosed
WO-1998057951-A1 NOVEL GUANIDINE MIMICS AS FACTOR Xa INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 1998-12-23 WO disclosed