SCHEMBL7369730

SCHEMBL7369730

CCCC(=O)CC(=O)NC

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.46
HDAC1 Q13547 4/20 0.46
HDAC2 Q92769 4/20 0.46
HDAC8 Q9BY41 4/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CTSD P07339 1/20 0.44
LMNA P02545 1/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
FFAR3 O14843 3/20 0.39
TSHR P16473 1/20 0.38
MCL1 Q07820 1/20 0.37
CASP2 P42575 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HAO1 Q9UJM8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2410237 0.85 HAO1 (0.47) LMNACES2CES1CASP2ALDH1A1
SCHEMBL14890831 0.83 HAO1 (0.45) LMNACES2CES1CASP2ALDH1A1
SCHEMBL21654407 0.83 HAO1 (0.55) CES2CES1TSHRALDH1A1HAO1
SCHEMBL13129296 0.82 LMNA (0.46) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL23281436 0.81 HAO1 (0.59) CES2CES1TSHRALDH1A1HAO1
SCHEMBL932939 0.81 HAO1 (0.59) CES2CES1TSHRALDH1A1HAO1
SCHEMBL8577435 0.81 HAO1 (0.59) CES2CES1TSHRALDH1A1HAO1
SCHEMBL8575600 0.81 HAO1 (0.59) CES2CES1TSHRALDH1A1HAO1
SCHEMBL42695 0.80
SCHEMBL1701664 0.80 CES2 (0.53) HDAC3HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230008875-A1 SUBSTITUTED LACTAMS SHOWING SEROTONIN 5-HT RECEPTOR ACTIVITY Sumitomo Pharma Co., Ltd. (JP) 2023-01-12 US disclosed
US-10988571-B2 Quorum sensing based polymer for stimulation of biofilms and related phenotypes, and synthesis process thereof FIB-SOL Life Technologies Private Limited (IN) 2021-04-27 US disclosed
US-10745401-B2 Condensed lactam derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-08-18 US disclosed
US-20200172543-A1 CONDENSED LACTAM DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2020-06-04 US disclosed
WO-2020022237-A1 FUSED RING LACTAM DERIVATIVES 大日本住友製薬株式会社 2020-01-30 WO disclosed
US-20200031989-A1 QUORUM SENSING BASED POLYMER FOR STIMULATION OF BIOFILMS AND RELATED PHENOTYPES, AND SYNTHESIS PROCESS THEREOF FIB-SOL Life Technologies Private Limited (IN) 2020-01-30 US disclosed
US-8199269-B2 Method for manufacturing thin film transistors HITACHI DISPLAYS, LTD. (JP) 2012-06-12 US disclosed
EP-1208208-B1 TRANSGENIC SYSTEMS FOR THE MANUFACTURE OF POLY(3-HYDROXY -BUTYRATE -CO -3- HYDROXYHEXANOATE) METABOLIX INC (US) 2009-06-17 EP disclosed
US-7455999-B2 Transgenic systems for the manufacture of poly (3-hydroxy-butyrate-co-3-hydroxyhexanoate) METABOLIX, INC. (US) 2008-11-25 US disclosed
EP-0808309-A1 IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS S-ADENOSYLMETHIONINE DECARBOXYLASE (=SAMDC) INHIBITORS Novartis AG (CH) 1997-11-26 EP disclosed
WO-1996022979-A1 IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS S-ADENOSYLMETHIONINE DECARBOXYLASE (=SAMDC) INHIBITORS NOVARTIS AG (CH) 1996-08-01 WO disclosed
WO-1996016980-A1 MORPHOLINOETHYLAMIDE DERIVATIVES NOVARTIS AG (CH) 1996-06-06 WO disclosed
EP-0708760-A1 CYCLIC HYDRAZINE COMPOUNDS Novartis AG (CH) 1996-05-01 EP disclosed
WO-1995002582-A1 CYCLIC HYDRAZINE COMPOUNDS CIBA-GEIGY AG (CH) 1995-01-26 WO disclosed
EP-0114059-B1 METHOD OF PREPARING A POLYAMIDE ACID COMPOSITION FOR PREPARING POLYIMIDE KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1989-06-14 EP disclosed
EP-0083690-B1 POLYAMIDE ACID COMPOSITION FOR PREPARING POLYIMIDE AND PROCESS FOR PREPARING POLYIMIDE FROM THE SAME KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1986-03-12 EP disclosed
US-4515915-A Polyamide acid composition for preparing polyimide KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1985-05-07 US disclosed
EP-0114059-A2 Method of preparing a polyamide acid composition for preparing polyimide KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1984-07-25 EP disclosed
US-4454276-A POT LIFE EXTENDING AGENT Kanegafuchi Chkagaku Kogyo Kabushiki Kaisha (JP) 1984-06-12 US disclosed
EP-0083690-A1 Polyamide acid composition for preparing polyimide and process for preparing polyimide from the same KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1983-07-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10988571-B2 Quorum sensing based polymer for stimulation of biofilms and related phenotypes, and synthesis process thereof PGLS, COASY, FDPS HDAC3 4261/4885HDAC1 4529/4885HDAC2 4821/4885
US-10745401-B2 Condensed lactam derivative PSEN1, GRIN1, HDAC1 HDAC3 123/4885HDAC1 3/4885HDAC2 15/4885
US-20230008875-A1 SUBSTITUTED LACTAMS SHOWING SEROTONIN 5-HT RECEPTOR ACTIVITY HTR1A, HTR5A, TPH1 HDAC3 2410/4885HDAC1 715/4885HDAC2 1320/4885
US-20200172543-A1 CONDENSED LACTAM DERIVATIVE PSEN1, GRIN1, HDAC1 HDAC3 123/4885HDAC1 3/4885HDAC2 15/4885
US-20200031989-A1 QUORUM SENSING BASED POLYMER FOR STIMULATION OF BIOFILMS AND RELATED PHENOTYPES, AND SYNTHESIS PROCESS THEREOF PGLS, COASY, FDPS HDAC3 4261/4885HDAC1 4529/4885HDAC2 4821/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.