SCHEMBL7370810

SCHEMBL7370810

Cc1ccc(-c2ccccc2C(=O)Nc2ccc(C(=O)N(C)c3ccccc3)c(Cl)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.52
POLB P06746 2/20 0.50
LMNA P02545 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
TP53 P04637 1/20 0.46
AVPR2 P30518 3/20 0.45
AVPR1A P37288 3/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HTT P42858 2/20 0.44
USP28 Q96RU2 1/20 0.44
GPR27 Q9NS67 1/20 0.44
DHODH Q02127 1/20 0.44
OPRL1 P41146 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8812976 0.90 MEN1 (0.51) L3MBTL1POLBLMNAMEN1KMT2A
SCHEMBL7377166 0.85 AVPR2 (0.48) L3MBTL1LMNAMEN1KMT2ATP53
SCHEMBL7371083 0.85 HTT (0.56) L3MBTL1POLBLMNAKMT2ATP53
SCHEMBL7378335 0.81 CHRNB2 (0.52) L3MBTL1POLBLMNAKMT2ATP53
SCHEMBL7517678 0.81 NPC1 (0.47) L3MBTL1POLBLMNAKMT2ATP53
SCHEMBL7376298 0.80 L3MBTL1 (0.48) L3MBTL1POLBLMNAKMT2ATP53
SCHEMBL7512593 0.80 CYP19A1 (0.45) L3MBTL1MEN1KMT2ATP53AVPR2
SCHEMBL7374840 0.79 PYGL (0.41) L3MBTL1LMNAMEN1KMT2AAVPR2
SCHEMBL7368408 0.79 HSD17B1 (0.58) L3MBTL1POLBLMNAKMT2ATP53
SCHEMBL7370671 0.78 GCGR (0.41) L3MBTL1POLBMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211242-B1 CARDIOVASCULAR DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-03 US disclosed
EP-0757670-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 1999-01-13 EP disclosed
WO-1995029152-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-02 WO disclosed