SCHEMBL7376137

SCHEMBL7376137

CCOC(=O)C(Sc1cccc(C)c1)C(=O)OCC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 2/20 0.44
HTT P42858 1/20 0.44
TP53 P04637 1/20 0.42
TDP1 Q9NUW8 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
HPGD P15428 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ALOX5 P09917 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369925 0.84 ALOX12 (0.44) ALDH1A1MAPTHTTGAANPSR1
SCHEMBL7371129 0.83 MTNR1B (0.54) ALDH1A1TDP1L3MBTL1TSHR
SCHEMBL8329718 0.83 PIN1 (0.50) ALDH1A1MAPTKDM4ETDP1HPGD
SCHEMBL6960077 0.80 KIF11 (0.40) HSD17B10ALOX5PPARGPPARALMNA
SCHEMBL7371798 0.79 EPHX1 (0.53) ALDH1A1MAPTKDM4EHTTTDP1
SCHEMBL15681420 0.75 TP53 (0.40) ALDH1A1MAPTTP53TDP1L3MBTL1
SCHEMBL12694091 0.75 ITGB3 (0.49) ALDH1A1MAPTGAANPSR1TSHR
SCHEMBL11599874 0.75 LMNA (0.41) MAPTHSD17B10ALOX5PPARGPPARA
SCHEMBL17785160 0.74 LMNA (0.50) ALDH1A1MAPTKDM4EHTTTP53
SCHEMBL19717928 0.73 KMT2A (0.45) ALDH1A1MAPTKDM4EHTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed