SCHEMBL7378633

SCHEMBL7378633

Cc1cnn(C(C)CCCc2ccccc2)c1N

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
POLB P06746 1/20 0.38
CYP2D6 P10635 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
MAOB P27338 2/20 0.37
DHFR P00374 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997571 0.82 ALDH1A1 (0.38) TSHRPOLBMAOB
SCHEMBL7893458 0.81 RIPK2 (0.46) TSHRCYP2D6PDE4APDE4BPDE4C
SCHEMBL27481625 0.81 L3MBTL1 (0.34) TSHRSIGMAR1MAOB
SCHEMBL7381725 0.79 PDE4A (0.39) PDE4APDE4BPDE4CPDE4D
SCHEMBL6996007 0.78 PDE4A (0.41) CYP2D6PDE4APDE4BPDE4CPDE4D
SCHEMBL7850685 0.78 NOS3 (0.40) POLBCYP2D6SIGMAR1NOS3NOS1
SCHEMBL7361207 0.70 KMT2A (0.45) TSHRPOLBCYP2D6PDE4APDE4B
SCHEMBL7843449 0.69 PDE4A (0.40) CYP2D6PDE4APDE4BPDE4CPDE4D
SCHEMBL7511580 0.69 LMNA (0.42) CYP2D6PDE4APDE4BPDE4CPDE4D
SCHEMBL27468086 0.69 GAA (0.52) TSHRPOLBDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973774-A1 1,5-DIHYDRO-PYRAZOLO 3,4-D]-PYRIMIDINONE DERIVATIVES BAYER AG (DE) 2000-01-26 EP disclosed
WO-1998040384-A1 1,5-DIHYDRO-PYRAZOLO[3,4-D]-PYRIMIDINONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1998-09-17 WO disclosed