SCHEMBL7850685

SCHEMBL7850685

Cc1nnn(C(C)CCCc2ccccc2)c1N

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
POLB P06746 1/20 0.38
CYP2D6 P10635 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
MAOB P27338 2/20 0.37
ATP4A P20648 1/20 0.36
ATP4B P51164 1/20 0.36
HDAC6 Q9UBN7 1/20 0.35
DAGLA Q9Y4D2 2/20 0.35
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361207 0.81 KMT2A (0.45) POLBCYP2D6DAGLA
SCHEMBL7511580 0.80 LMNA (0.42) CYP2D6DAGLA
SCHEMBL7843449 0.80 PDE4A (0.40) CYP2D6DAGLA
SCHEMBL7378633 0.78 TSHR (0.49) NOS3NOS1NOS2POLBCYP2D6
SCHEMBL6997571 0.71 ALDH1A1 (0.38) POLBMAOB
SCHEMBL2883347 0.70 ADORA3 (0.42) POLBSIGMAR1
SCHEMBL6996007 0.70 PDE4A (0.41) CYP2D6
SCHEMBL27481625 0.70 L3MBTL1 (0.34) SIGMAR1MAOB
SCHEMBL7893458 0.70 RIPK2 (0.46) CYP2D6
SCHEMBL27468086 0.69 GAA (0.52) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107968-A2 DIHYDRO-[1,2,3]TRIAZOLO-[4,5-D]PYRIMIDIN-7-ONE BAYER AG (DE) 2001-06-20 EP disclosed
WO-2000012504-A2 DIHYDRO-[1,2,3]TRIAZOLO-[4,5-D]PYRIMIDIN-7-ONE BAYER AKTIENGESELLSCHAFT (DE) 2000-03-09 WO disclosed