SCHEMBL7410782

SCHEMBL7410782

CNC(=O)N(CC(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)CCc1ccccc1)C(C)C)Cc1ccncc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.48
BACE1 P56817 4/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
MMP9 P14780 4/20 0.37
MMP8 P22894 2/20 0.37
ELANE P08246 1/20 0.36
MMP1 P03956 3/20 0.36
MMP2 P08253 2/20 0.36
MMP3 P08254 2/20 0.36
MMP7 P09237 1/20 0.36
MMP14 P50281 1/20 0.36
HTRA1 Q92743 1/20 0.36
HRH1 P35367 3/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7413833 0.92 CASP1 (0.47) CASP1ALDH1A1CYP3A4MMP9MMP8
SCHEMBL7415944 0.89 CASP1 (0.47) CASP1ALDH1A1ELANECA2
SCHEMBL7419381 0.79 CASP1 (0.48) CASP1ELANEMMP3CA2
SCHEMBL7415572 0.77 CASP1 (0.54) CASP1BACE1HTRA1
SCHEMBL9578947 0.76 CA2 (0.47) CASP1HTRA1CA2
SCHEMBL7423302 0.75 CASP1 (0.52) CASP1ELANEHTRA1
SCHEMBL7419148 0.73 CTSL (0.49) CASP1CYP3A4ELANE
SCHEMBL7410781 0.73 CASP1 (0.52) CASP1ELANEMMP3CA2
SCHEMBL7418881 0.73 ALDH1A1 (0.46) BACE1ALDH1A1CYP3A4MMP9MMP8
SCHEMBL9579040 0.72 CASP3 (0.46) CASP1ELANECA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO claimed
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed