SCHEMBL7413833

SCHEMBL7413833

CNC(=O)N(CC(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)CCc1ccccc1)C(C)C)Cc1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.47
MMP12 P39900 2/20 0.42
ALDH1A1 P00352 2/20 0.39
ELANE P08246 1/20 0.39
LMNA P02545 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38
ADRA1B P35368 1/20 0.38
DRD3 P35462 1/20 0.38
HTR2B P41595 1/20 0.38
HTR5A P47898 1/20 0.38
CTSD P07339 3/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410782 0.92 CASP1 (0.48) CASP1ALDH1A1ELANEMMP1MMP3
SCHEMBL7415944 0.88 CASP1 (0.47) CASP1ALDH1A1ELANECTSD
SCHEMBL7419148 0.80 CTSL (0.49) CASP1ELANECTSLCTSBCYP3A4
SCHEMBL7415572 0.75 CASP1 (0.54) CASP1CTSDCTSB
SCHEMBL9578947 0.74 CA2 (0.47) CASP1CTSD
SCHEMBL7423302 0.74 CASP1 (0.52) CASP1ELANECTSDCTSLCTSB
SCHEMBL7414554 0.73 CMA1 (0.40) MMP12ELANECTSLCTSBMMP9
SCHEMBL7419381 0.73 CASP1 (0.48) CASP1ELANECTSDCTSLCTSB
SCHEMBL7410781 0.72 CASP1 (0.52) CASP1ELANECTSDCTSLCTSB
SCHEMBL9579040 0.71 CASP3 (0.46) CASP1ELANECTSDCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO claimed
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed