SCHEMBL7414554

SCHEMBL7414554

CC(C)[C@@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)CCc1ccccc1)N(C(=O)CN)C(=O)NCc1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 2/20 0.40
CTRC Q99895 2/20 0.40
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ELANE P08246 1/20 0.39
CYP3A4 P08684 2/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MMP12 P39900 2/20 0.38
KLKB1 P03952 3/20 0.38
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37
REN P00797 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418881 0.92 ALDH1A1 (0.46) CMA1CTRCMMP9MMP8ELANE
SCHEMBL7414431 0.88 TSHR (0.47) CYP1A2RENSMN1; SMN2
SCHEMBL7413833 0.73 CASP1 (0.47) MMP9MMP8ELANECYP3A4CTSL
SCHEMBL7419148 0.72 CTSL (0.49) ELANECYP3A4CTSLCTSBREN
SCHEMBL9578947 0.68 CA2 (0.47) CYP1A2RENSMN1; SMN2
SCHEMBL7410782 0.67 CASP1 (0.48) MMP9MMP8ELANECYP3A4
SCHEMBL7415572 0.67 CASP1 (0.54) CTSB
SCHEMBL7270435 0.66 L3MBTL1 (0.47) L3MBTL1CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL7419381 0.65 CASP1 (0.48) CTRCELANECTSLCTSBREN
SCHEMBL7415944 0.64 CASP1 (0.47) ELANECYP1A2KMT2ARENSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO claimed
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed