SCHEMBL7434827

SCHEMBL7434827

CCCCSc1ccc2c(c1)OCC(C(=O)C1COc3cc(SCCCC)ccc3O1)O2

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.45
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 1/20 0.36
THRB P10828 2/20 0.36
ITGB2 P05107 1/20 0.35
ICAM1 P05362 1/20 0.35
ITGAL P20701 1/20 0.35
HSD17B10 Q99714 3/20 0.35
TP53 P04637 1/20 0.35
PKM P14618 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434823 0.80 AR (0.37) HPGDALDH1A1KDM4ENPC1RAB9A
SCHEMBL7434686 0.80 NPC1 (0.42) HPGDALDH1A1MAPTNPC1RAB9A
SCHEMBL7427958 0.80 TSHR (0.47) HPGDMAPTKDM4ERAB9ASMN1; SMN2
SCHEMBL7437379 0.76 MAOA (0.35) HPGDALDH1A1MAPTKDM4ENPC1
SCHEMBL7440246 0.74 HPGD (0.44) HPGDALDH1A1KDM4EKMT2ATHRB
SCHEMBL7446273 0.73 HPGD (0.44) HPGDALDH1A1MAPTKDM4ENPC1
SCHEMBL7437345 0.72 RAB9A (0.50) HPGDALDH1A1MAPTNPC1RAB9A
SCHEMBL14501846 0.72 LMNA (0.44) HPGDALDH1A1MAPTKDM4ENPC1
SCHEMBL14501849 0.72 LMNA (0.44) HPGDALDH1A1MAPTKDM4ENPC1
SCHEMBL10993172 0.70 ALDH1A1 (0.36) ALDH1A1KDM4ENPC1RAB9ATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed