SCHEMBL7440246

SCHEMBL7440246

CCCCS(=O)(=O)c1ccc2c(c1)OCC(C(=O)C1COc3cc(S(=O)(=O)CCCC)ccc3O1)O2

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.44
POLB P06746 3/20 0.44
TP53 P04637 1/20 0.41
GLA P06280 1/20 0.40
LMNA P02545 3/20 0.40
CYP2C9 P11712 1/20 0.39
THRB P10828 3/20 0.39
PNMT P11086 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440239 0.81 PNMT (0.39) HPGDPOLBLMNACYP2C9THRB
SCHEMBL7437881 0.80 ALDH1A1 (0.49) POLBTP53GLALMNAL3MBTL1
SCHEMBL7426673 0.80 HPGD (0.48) HPGDTHRBALDH1A1MEN1KMT2A
SCHEMBL7435505 0.78 PNMT (0.36) HPGDPOLBLMNATHRBPNMT
SCHEMBL7427958 0.76 TSHR (0.47) HPGDTHRBKDM4EMEN1KMT2A
SCHEMBL7446273 0.75 HPGD (0.44) HPGDPOLBGLAALDH1A1KDM4E
SCHEMBL7434827 0.74 HPGD (0.45) HPGDTP53THRBALDH1A1KDM4E
SCHEMBL10989168 0.72 THRB (0.36) POLBTHRBPNMT
SCHEMBL7437345 0.71 RAB9A (0.50) HPGDPOLBL3MBTL1ALDH1A1
SCHEMBL7435716 0.71 PNMT (0.33) HPGDPOLBTHRBPNMTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed