SCHEMBL744198

SCHEMBL744198

C[C@H]1C[C@H](O)CN1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.48
PIK3CD O00329 5/20 0.41
DPP4 P27487 7/20 0.37
DPP8 Q6V1X1 7/20 0.37
DPP9 Q86TI2 7/20 0.37
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
FAP Q12884 1/20 0.35
RIPK1 Q13546 1/20 0.35
GAA P10253 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1923005 1.00 ATM (0.48) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL17760540 1.00 ATM (0.48) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL4531927 1.00 ATM (0.48) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL3673559 1.00 ATM (0.48) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL746205 1.00 ATM (0.48) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL25286686 1.00 ATM (0.48) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL5795993 1.00 ATM (0.48) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL418951 0.82 ATM (0.59) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL16751022 0.82 ATM (0.59) ATMPIK3CDDPP4DPP8DPP9
SCHEMBL17511112 0.80 ATM (0.42) ATMPIK3CDDPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240238300-A1 TREATMENT METHODS FOR SUBJECTS WITH CANCER HAVING AN ABERRATION IN EGFR AND/OR HER2 TAIHO PHARMACEUTICAL CO., LTD. (JP) 2024-07-18 US disclosed
EP-4359082-A1 HER2 MUTATION INHIBITORS Array BioPharma Inc. (US) 2024-05-01 EP disclosed
US-20240067632-A1 WEE1 Degrading Compounds and Uses Thereof BRISTOL-MYERS SQUIBB COMPANY (US) 2024-02-29 US disclosed
US-11878976-B2 FGFR3 inhibitor compounds ELI LILLY AND COMPANY (US) 2024-01-23 US disclosed
EP-3909584-B1 PYRIMIDINE COMPOUND OR SALT THEREOF TAIHO PHARMACEUTICAL CO LTD (JP) 2023-12-13 EP disclosed
US-20230331730-A1 CRYSTAL OF PYRIMIDINE COMPOUND TAIHO PHARMACEUTICAL CO., LTD. (JP) 2023-10-19 US disclosed
US-20230285397-A1 EGFR INHIBITOR TAIHO PHARMACEUTICAL CO., LTD. (JP) 2023-09-14 US disclosed
US-20230255972-A1 PYRIMIDINE COMPOUND-CONTAINING COMBINATION TO BE USED IN TUMOR TREATMENT TAIHO PHARMACEUTICAL CO., LTD. (JP) 2023-08-17 US disclosed
US-11696917-B2 Agent enhancing antitumor effect using pyrazolo[3,4-d]pyrimidine compound TAIHO PHARMACEUTICAL CO., LTD. (JP) 2023-07-11 US disclosed
US-20230203060-A1 FUSED TRICYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF GENFLEET THERAPEUTICS (SHANGHAI) INC. (CN) 2023-06-29 US disclosed
EP-2431357-A2 3-Aminopyrrolidine Derivatives as Modulators of Chemokine Receptors Incyte Corporation (US) 2012-03-21 EP disclosed
US-20110251168-A1 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE CORPORATION 2011-10-13 US disclosed
US-7985730-B2 3-aminopyrrolidine derivatives as modulators of chemokine receptors INCYTE CORPORATION (US) 2011-07-26 US disclosed
US-7834021-B2 3-aminopyrrolidine derivatives as modulators of chemokine receptors INCYTE CORPORATION (US) 2010-11-16 US disclosed
US-20090264431-A1 NOVEL CATHEPSIN C INHIBITORS AND THEIR USE GLAXO GROUP LIMITED (GB) 2009-10-22 US disclosed
US-20090247474-A1 3-Aminopyrrolidine Derivatives As Modulators Of Chemokine Receptors INCYTE CORPORATION 2009-10-01 US disclosed
EP-1565436-A4 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE CORP (US) 2007-07-18 EP disclosed
US-20060252751-A1 3-Aminopyrrolidine derivaties as modulators of chemokine receptors INCYTE HOLDINGS CORPORATION 2006-11-09 US disclosed
EP-1565436-A2 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE CORPORATION (US) 2005-08-24 EP disclosed
WO-2004050024-A2 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS INCYTE CORPORATION (US) 2004-06-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230331730-A1 CRYSTAL OF PYRIMIDINE COMPOUND DPYD, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, UMPS ATM 1368/4885PIK3CD 2349/4885DPP4 399/4885
US-20060252751-A1 3-Aminopyrrolidine derivaties as modulators of chemokine receptors CCR2, CXCR3, CCR5 ATM 2071/4885PIK3CD 3629/4885DPP4 2633/4885
US-20090264431-A1 NOVEL CATHEPSIN C INHIBITORS AND THEIR USE CTSB, CTSS, CTSF ATM 4495/4885PIK3CD 3793/4885DPP4 701/4885
US-11696917-B2 Agent enhancing antitumor effect using pyrazolo[3,4-d]pyrimidine compound ZYX, DPYD, ZFX ATM 2546/4885PIK3CD 1805/4885DPP4 268/4885
US-20230285397-A1 EGFR INHIBITOR EGFR, ERBB2, ERBB4 ATM 1416/4885PIK3CD 706/4885DPP4 1636/4885
US-11878976-B2 FGFR3 inhibitor compounds FGFR3, FGFR1, FGFR2 ATM 1958/4885PIK3CD 2062/4885DPP4 3146/4885
US-20240238300-A1 TREATMENT METHODS FOR SUBJECTS WITH CANCER HAVING AN ABERRATION IN EGFR AND/OR HER2 EGFR, ERBB2, ERBB3 ATM 139/4885PIK3CD 657/4885DPP4 1413/4885
US-20230255972-A1 PYRIMIDINE COMPOUND-CONTAINING COMBINATION TO BE USED IN TUMOR TREATMENT TYMP, DPYD, TYMS ATM 1711/4885PIK3CD 1880/4885DPP4 2584/4885
US-20230203060-A1 FUSED TRICYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF KRAS, NRAS, TP53 ATM 1709/4885PIK3CD 46/4885DPP4 2706/4885
US-20090247474-A1 3-Aminopyrrolidine Derivatives As Modulators Of Chemokine Receptors CCR2, CXCR3, CCR5 ATM 2379/4885PIK3CD 3597/4885DPP4 2716/4885
US-20240067632-A1 WEE1 Degrading Compounds and Uses Thereof WEE1, WEE2, PPME1 ATM 444/4885PIK3CD 1035/4885DPP4 3709/4885
US-20110251168-A1 3-AMINOPYRROLIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTORS CCR2, CXCR3, CCR5 ATM 2379/4885PIK3CD 3597/4885DPP4 2716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.