SCHEMBL7445935

SCHEMBL7445935

COc1cc(OC2CCCN(OC(C)(C)C)C2=C=O)ccc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM2B Q8NHM5 3/20 0.39
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
HIF1A Q16665 1/20 0.36
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
OXTR P30559 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
PARP15 Q460N3 1/20 0.35
PARP10 Q53GL7 1/20 0.35
ATM Q13315 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3563776 0.73 GRIK1 (0.43) KDM2BALDH1A1RAB9AMEN1KMT2A
SCHEMBL7404006 0.71 PDE4B (0.52) KDM2BHIF1A
SCHEMBL7355186 0.70 GPR119 (0.54) ALDH1A1MEN1KMT2ATSHR
SCHEMBL8902641 0.69 HIF1A (0.63) ALDH1A1RAB9AHIF1AMEN1KMT2A
SCHEMBL7402370 0.68 PDE4B (0.52) ALDH1A1MEN1KMT2ATSHR
SCHEMBL7356525 0.67 HIF1A (0.34) KDM2BALDH1A1RAB9AHIF1AOXTR
SCHEMBL3823895 0.67 RAB9A (0.38) KDM2BALDH1A1RAB9AMEN1KMT2A
SCHEMBL8094956 0.67 LIPG (0.38)
SCHEMBL2588369 0.67 ALDH1A1 (0.56) ALDH1A1RAB9AMEN1KMT2AAKR1C3
SCHEMBL8665462 0.67 OXTR (0.55) ALDH1A1HIF1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714299-A4 1996-07-10 EP disclosed
EP-0714299-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO. INC. (US) 1996-06-05 EP disclosed
WO-1995002405-A1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1995-01-26 WO disclosed