SCHEMBL7465748

SCHEMBL7465748

COc1ccc(/C=C/C(=O)N2C[C@@H](CCl)c3c2cc(O)c2[nH]c(C(F)(F)F)c(C(=O)O)c32)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
HPGD P15428 3/20 0.37
GAA P10253 3/20 0.37
LMNA P02545 2/20 0.37
GPR183 P32249 2/20 0.36
MAPT P10636 1/20 0.35
ACHE P22303 2/20 0.34
SLC5A1 P13866 1/20 0.34
SLC5A2 P31639 1/20 0.34
BCHE P06276 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
MAOB P27338 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7465921 1.00 ALDH1A1 (0.37) ALDH1A1HPGDGAALMNAGPR183
SCHEMBL7470246 0.82 HRH3 (0.34) ALDH1A1HPGD
SCHEMBL7474728 0.79 MGLL (0.35) ACHENPC1RAB9ACYP1A2CYP2D6
SCHEMBL6851179 0.79 ADH1A (0.35)
SCHEMBL7465950 0.76 AKR1C3 (0.39) ALDH1A1HPGDLMNAMAPTNPC1
SCHEMBL7470331 0.75 LMNA (0.36) ALDH1A1LMNAMAPTNPC1RAB9A
SCHEMBL7463040 0.74 ADH1A (0.33) ACHE
SCHEMBL7465517 0.74 KDM4E (0.36) ALDH1A1GAAMAPTACHENPC1
SCHEMBL6851145 0.73 ADH1A (0.39) ALDH1A1HPGDGPR183MAPTNPC1
SCHEMBL7474788 0.73 P4HB (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656360-B1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2002-11-20 EP disclosed
US-5629430-A ANTICARCINOGENIC AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-05-13 US disclosed
EP-0656360-A1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1995-06-07 EP disclosed