SCHEMBL7470246

SCHEMBL7470246

COc1ccc2oc(C(=O)N3C[C@@H](CCl)c4c3cc(O)c3[nH]c(C(F)(F)F)c(C(=O)O)c43)cc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.34
PIM1 P11309 1/20 0.34
TAS1R3 Q7RTX0 8/20 0.34
TAS1R1 Q7RTX1 8/20 0.34
ALDH1A1 P00352 4/20 0.33
HTR1A P08908 2/20 0.32
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
DRD3 P35462 2/20 0.32
KDM4E B2RXH2 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA3 P07451 1/20 0.32
HPGD P15428 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7474728 0.94 MGLL (0.35) HRH3
SCHEMBL7465517 0.87 KDM4E (0.36) TAS1R3TAS1R1ALDH1A1HTR1ADRD2
SCHEMBL7470331 0.86 LMNA (0.36) ALDH1A1DRD2DRD3KDM4ECA12
SCHEMBL7463040 0.85 ADH1A (0.33)
SCHEMBL13401627 0.85 TAS1R3 (0.37) TAS1R3TAS1R1HTR1ADRD2HTR2A
SCHEMBL7474788 0.84 P4HB (0.34)
SCHEMBL7465921 0.82 ALDH1A1 (0.37) ALDH1A1HPGD
SCHEMBL7465748 0.82 ALDH1A1 (0.37) ALDH1A1HPGD
SCHEMBL7464956 0.82 KDM4E (0.35) ALDH1A1KDM4E
SCHEMBL16349649 0.80 HRH4 (0.34) HRH3ALDH1A1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656360-B1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2002-11-20 EP disclosed
US-5629430-A ANTICARCINOGENIC AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-05-13 US disclosed
EP-0656360-A1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1995-06-07 EP disclosed