SCHEMBL7470869

SCHEMBL7470869

NC(=O)CC(Br)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.51
CYP2D6 P10635 2/20 0.48
CYP1A2 P05177 1/20 0.48
PKM P14618 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
SLC6A3 Q01959 3/20 0.47
DRD3 P35462 2/20 0.47
LMNA P02545 2/20 0.47
MAPK1 P28482 2/20 0.47
ADORA3 P0DMS8 1/20 0.47
EDNRB P24530 1/20 0.47
MC4R P32245 1/20 0.47
MC3R P41968 1/20 0.47
DRD2 P14416 1/20 0.47
GABBR2 O75899 1/20 0.46
GABBR1 Q9UBS5 1/20 0.46
EPHX1 P07099 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL777871 0.83 GABBR2 (0.53) CYP2C19CYP2D6CES2CES1LMNA
SCHEMBL11017601 0.82 SLC6A3 (0.50) CYP2C19CYP2D6CYP1A2PKMSMN1; SMN2
SCHEMBL1383474 0.80 CYP2C19 (0.67) CYP2C19CYP2D6CYP1A2PKMSMN1; SMN2
SCHEMBL2655629 0.79 CES2 (0.48) CYP2D6CES2CES1LMNAMAPK1
SCHEMBL22319291 0.79 CES2 (0.48) CYP2D6CES2CES1LMNAMAPK1
Hydrochloric Acid SCHEMBL29096814 0.78 CYP2C19 (0.65) CYP2C19CYP2D6CYP1A2PKMSMN1; SMN2
SCHEMBL9105247 0.78 ALDH1A1 (0.63) CYP2C19CYP2D6CYP1A2PKMSMN1; SMN2
Hydrochloric Acid SCHEMBL5011439 0.78 CYP2C19 (0.65) CYP2C19CYP2D6CYP1A2PKMSMN1; SMN2
SCHEMBL7757013 0.78 TSHR (0.57) CYP2C19CYP1A2SMN1; SMN2NPSR1CES2
SCHEMBL1847912 0.77 BCAT2 (0.58) CYP2C19CYP2D6CYP1A2PKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103739547-B The synthetic method of 2-[6-methoxyl group-3-(2,3-dichlorophenyl) methyl-4-oxo-Isosorbide-5-Nitrae-dihydro-1 (4H)-quinolyl] acetic acid SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2015-09-02 CN disclosed
CN-103739547-A Synthesis method of 2-[6-methoxy-3-(2,3-dichlorophenyl)methyl-4-oxo-1,4-dihydro-1(4H)-quinolyl] acetic acid UNIV SHENYANG PHARMACEUTICAL 2014-04-23 CN disclosed
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
CN-1292697-A Anti-viral compound LILLY CO ELI (US) 2001-04-25 CN disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed