SCHEMBL74997

SCHEMBL74997

COc1ccc(S(=O)(=O)Cl)c(OC)c1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.68
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52
GAA P10253 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
ALPL P05186 2/20 0.48
ALDH1A1 P00352 2/20 0.47
CYP19A1 P11511 1/20 0.47
CYP1A1 P04798 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP1B1 Q16678 2/20 0.46
CYP3A4 P08684 1/20 0.46
TP53 P04637 1/20 0.45
GFER P55789 1/20 0.45
MMP7 P09237 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29482639 1.00 TRPV4 (0.68) TRPV4CA12CA1CA2CA7
SCHEMBL29482636 0.85 L3MBTL1 (0.64) TRPV4CA12CA1CA2CA7
SCHEMBL407215 0.85 L3MBTL1 (0.64) TRPV4CA12CA1CA2CA7
SCHEMBL2494884 0.83 TRPV4 (0.49) TRPV4CA12CA1CA2CA7
SCHEMBL2497225 0.83 TRPV4 (0.49) TRPV4CA12CA1CA2CA7
SCHEMBL2502219 0.83 TRPV4 (0.57) TRPV4GAAALPL
SCHEMBL2498920 0.83 TRPV4 (0.57) TRPV4GAAALPLMMP7
SCHEMBL31518304 0.83 TRPV4 (0.57) TRPV4CA1CA2CA9L3MBTL1
SCHEMBL2719702 0.82 CA12 (0.54) TRPV4CA12CA1CA2CA7
SCHEMBL533956 0.81 TRPV4 (0.68) TRPV4CA1CA2CA9GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 388 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104678028-A Pretreatment and detection method for biogen amine neurotransmitter and detection kit INST PHARM & TOXICOLOGY AMMS 2015-06-03 CN claimed
EP-4743176-A1 DEUTERATED 1,3 DIHYDRO -2H-INDOLE-2-ONE DERIVATIVES HMNC Holding GmbH (DE) 2026-05-20 EP disclosed
EP-4168399-B1 COMPOUNDS AND THEIR USES AS MIF INHIBITORS NANJING IMMUNOPHAGE BIOMEDICAL CO LTD (CN) 2026-04-01 EP disclosed
US-20260062393-A1 Compounds CTXT PTY LTD (AU) 2026-03-05 US disclosed
US-12479842-B2 Pyrido[3,2-d]pyrimidine compounds uses thereof for treating a proliferative disease UNIVERSITE DE MONTREAL (CA) 2025-11-25 US disclosed
US-20250270207-A1 PYRIDO[3,2-D]PYRIMIDINE COMPOUNDS USES THEREOF FOR TREATING A PROLIFERATIVE DISEASE UNIVERSITE DE MONTREAL (CA) 2025-08-28 US disclosed
US-12365655-B2 Compounds CTXT PTY LTD (AU) 2025-07-22 US disclosed
US-20250122182-A1 MYST Inhibitors Isosterix, Inc. 2025-04-17 US disclosed
CN-119462588-A Flavone derivative containing sulfonamide structure and preparation method and application thereof 上海中医药大学附属曙光医院 2025-02-18 CN disclosed
US-20250034117-A1 Deuterated 1,3 Dihydro -2H-indole-2-one derivatives HMNC Holding GmbH (DE) 2025-01-30 US disclosed
US-5481005-A N-sulfonylindoline derivatives, their preparation and the pharmaceutical compositions in which they are present SANOFI (FR) 1996-01-02 US disclosed
CN-1107467-A 1-benzenesulfonyl-1,3-dihydro-indol-2-one derivatives, their preparation and pharmaceutical compositions in which they are present SANOFI SA (FR) 1995-08-30 CN disclosed
US-5397801-A Affinity for vasopressin and ocytocin receptors; disorders of nervous, cardiovascular and gastrointestinal systems SANOFI (FR) 1995-03-14 US disclosed
US-5338755-A Have affinity for vasopressin and ocytocin receptors; intermediates for drugs that act on central nervous system ELF SANOFI (FR) 1994-08-16 US disclosed
US-4714700-A TRANQUILIZERS, ANXIOLYTIC AGENTS CHOAY S.A. (FR) 1987-12-22 US disclosed
US-4618459-A INTERMEDIATES FOR BENZENESULFONAMIDE DERIVATIVES; ANTIDEPRESSANTS CHOAY S.A. (FR) 1986-10-21 US disclosed
US-4457875-A ANTIDEPRESSANTS, TRANQUILIZERS CHOAY S.A. (FR) 1984-07-03 US disclosed
EP-0056274-B1 INDOLE DERIVATIVES AND A METHOD FOR PRODUCTION OF PEPTIDES Takeda Chemical Industries, Ltd. (JP) 1984-05-09 EP disclosed
US-4416820-A Indole derivatives and a method for production of peptides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1983-11-22 US disclosed
EP-0056274-A1 Indole derivatives and a method for production of peptides Takeda Chemical Industries, Ltd. (JP) 1982-07-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250270207-A1 PYRIDO[3,2-D]PYRIMIDINE COMPOUNDS USES THEREOF FOR TREATING A PROLIFERATIVE DISEASE BRAF, NRAS, KRAS TRPV4 3761/4885CA12 4806/4885CA1 4840/4885
US-20260062393-A1 Compounds SCN2B, ABCB11, SCN1B TRPV4 1449/4885CA12 906/4885CA1 1778/4885
US-20250034117-A1 Deuterated 1,3 Dihydro -2H-indole-2-one derivatives IDO1, IDO2, TPH1 TRPV4 1518/4885CA12 1624/4885CA1 1367/4885
US-12479842-B2 Pyrido[3,2-d]pyrimidine compounds uses thereof for treating a proliferative disease BRAF, NRAS, DPYD TRPV4 3686/4885CA12 4810/4885CA1 4841/4885
US-20250122182-A1 MYST Inhibitors MNAT1, SUGT1, ACAT2 TRPV4 4752/4885CA12 4788/4885CA1 4866/4885
US-12365655-B2 Compounds SLC10A1, ABCB11, PCSK9 TRPV4 909/4885CA12 365/4885CA1 881/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.