SCHEMBL7517843

SCHEMBL7517843

CCc1cc(CC[Si](C)(C)c2ccc(N(C)C)cc2)cc(CC)c1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 2/20 0.36
G6PD P11413 1/20 0.36
CCR6 P51684 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
PSMB5 P28074 1/20 0.35
MAPT P10636 3/20 0.34
DHFR P00374 2/20 0.33
MAPK1 P28482 2/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
NPC1 O15118 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7517862 0.82 AKT1 (0.34) CALM1PSMB5MAPTMAPK1ALDH1A1
SCHEMBL9187478 0.73 DHFR (0.41) DHFRMAPK1GABRA1GABRB2ALDH1A1
SCHEMBL5692252 0.73 DHFR (0.41) DHFRMAPK1GABRA1GABRB2ALDH1A1
SCHEMBL5692097 0.72 ALOX5 (0.39) MAPTDHFRGABRA1GABRB2NPC1
SCHEMBL14370359 0.71 DHFR (0.40) DHFRGABRA1GABRB2CYP3A4BACE1
SCHEMBL5692247 0.70 TYR (0.37) MAPTMAPK1ALDH1A1CYP3A4NPC1
SCHEMBL28745704 0.70 GABRA1 (0.37) DHFRMAPK1GABRA1GABRB2ALDH1A1
SCHEMBL7522609 0.70 CALM1 (0.33) CALM1MAPTALDH1A1HDAC1HDAC2
SCHEMBL7521009 0.70 VCAM1 (0.37) CALM1GAA
SCHEMBL8385660 0.69 ALOX5 (0.37) MAPTDHFRNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
EP-0900225-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1999-03-10 EP disclosed
WO-1997041129-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-11-06 WO disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed