SCHEMBL7533413

SCHEMBL7533413

O=[C]Nc1cccc(CCl)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
RAPGEF4 Q8WZA2 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTR6 P50406 2/20 0.33
MAPT P10636 2/20 0.32
GAA P10253 1/20 0.32
F12 P00748 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27362602 0.81 HTR6 (0.50) TSHRHTR6
SCHEMBL1188671 0.81 RAPGEF4 (0.53) RAPGEF4MAPTGAASIGMAR1MEN1
SCHEMBL630874 0.79 MEN1 (0.42) NPSR1MAPTGAAMEN1ALDH1A1
SCHEMBL10388288 0.78 SIGMAR1 (0.47) RAPGEF4HTR6MAPTGAASIGMAR1
SCHEMBL7528041 0.75 CA1 (0.39)
SCHEMBL7351050 0.75 HDAC4 (0.44) HTR6
SCHEMBL5543430 0.74 LPL (0.47)
SCHEMBL57436 0.74 MEN1 (0.53) TSHRMAPTGAAMEN1ALDH1A1
SCHEMBL16230165 0.74 TSHR (0.42) TSHRRAPGEF4NPSR1HTR6MAPT
SCHEMBL6535170 0.73 ALDH1A1 (0.48) TSHRNPSR1HTR6MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed