SCHEMBL7537677

SCHEMBL7537677

Cc1csc(C(=O)Nc2ccc(Cl)cc2)c1NS(=O)(=O)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.59
MEN1 O00255 2/20 0.59
GPR27 Q9NS67 10/20 0.55
KDM4E B2RXH2 1/20 0.51
GAA P10253 1/20 0.51
MAPT P10636 1/20 0.51
F10 P00742 1/20 0.49
GRM4 Q14833 1/20 0.49
AVPR2 P30518 2/20 0.48
ENPP3 O14638 1/20 0.47
ENPP1 P22413 1/20 0.47
IDH1 O75874 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7561597 0.88 GPR27 (0.54) KMT2AMEN1GPR27KDM4EGAA
SCHEMBL7537898 0.85 GPR27 (0.54) KMT2AMEN1GPR27GAAMAPT
SCHEMBL7539025 0.79 MEN1 (0.62) KMT2AMEN1GPR27KDM4EMAPT
SCHEMBL7539008 0.74 LMNA (0.60) KMT2AMEN1GPR27KDM4EGAA
SCHEMBL7531362 0.74 KMT2A (0.62) KMT2AMEN1GPR27KDM4EGAA
SCHEMBL7530840 0.74 MEN1 (0.62) KMT2AMEN1GPR27KDM4EGRM4
SCHEMBL7537998 0.73 PGR (0.55) KMT2AMEN1GPR27KDM4EGRM4
SCHEMBL7534188 0.73 F10 (0.58) KMT2AMEN1KDM4EMAPTF10
SCHEMBL27180378 0.71 GPR27 (0.72) KMT2AMEN1GPR27KDM4EMAPT
SCHEMBL17593181 0.71 KMT2A (0.92) KMT2AMEN1GPR27MAPTGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002028353-A2 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-11 WO disclosed