SCHEMBL7556078

SCHEMBL7556078

Cc1c(C(CCCl)C(=O)C2CCCC2)ccc2[nH]c(CNc3ccc(C#N)cc3)nc12

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DGAT2 Q96PD7 2/20 0.35
TGFBR1 P36897 3/20 0.33
IDH1 O75874 2/20 0.33
PAX8 Q06710 1/20 0.32
HCRTR1 O43613 2/20 0.31
HCRTR2 O43614 2/20 0.31
ALDH1A1 P00352 2/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
MLLT1 Q03111 1/20 0.31
CTSC P53634 1/20 0.31
RORC P51449 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448201 0.70 EPHX2 (0.39) DGAT2TGFBR1IDH1ALDH1A1NPC1
SCHEMBL7423476 0.69 ITK (0.47) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL6455288 0.69 MLLT1 (0.33) DGAT2TGFBR1MLLT1
SCHEMBL7449699 0.68 MLLT1 (0.38) DGAT2TGFBR1IDH1ALDH1A1NPC1
SCHEMBL7448750 0.68 PDE2A (0.36) TGFBR1IDH1PAX8ALDH1A1NPC1
SCHEMBL7449392 0.67 NPC1 (0.34) TGFBR1PAX8ALDH1A1NPC1LMNA
SCHEMBL7445307 0.67 TGFBR1 (0.40) TGFBR1IDH1ALDH1A1NPC1LMNA
SCHEMBL7556081 0.67 DGAT2 (0.38) DGAT2ALDH1A1NPC1MLLT1KDM4E
SCHEMBL16268845 0.67 TGFBR1 (0.41) TGFBR1IDH1ALDH1A1NPC1LMNA
SCHEMBL7447468 0.66 TGFBR1 (0.46) TGFBR1IDH1ALDH1A1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed