SCHEMBL760695

SCHEMBL760695

Oc1cc(F)c(OC(F)(F)F)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
AURKA O14965 1/20 0.35
TPX2 Q9ULW0 1/20 0.35
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
EPHX2 P34913 1/20 0.34
BACE1 P56817 1/20 0.32
GPR84 Q9NQS5 1/20 0.32
PDE2A O00408 1/20 0.32
PTGS1 P23219 2/20 0.31
KIF11 P52732 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
FFAR1 O14842 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
GPR3 P46089 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29320324 0.87 AURKA (0.41) CA12CA1CA9TDP1AURKA
SCHEMBL31256373 0.86 ALOX5 (0.33) TAAR1CA12CA1CA9AURKA
SCHEMBL18559875 0.80 TAAR1 (0.33) TAAR1CA12CA1CA9TDP1
SCHEMBL12736297 0.80 GPR3 (0.33) EPHX2PDE2AGPR3
SCHEMBL23484287 0.78 TDP1 (0.48) CA12CA1CA9TDP1AURKA
SCHEMBL6558034 0.76 MAPT (0.36) MAPTEPHX2PDE2AGPR3
SCHEMBL3683516 0.76 GPR3 (0.31) EPHX2GPR3
SCHEMBL7723333 0.76 GPR3 (0.31) EPHX2PDE2AGPR3
SCHEMBL10052628 0.76 ACHE (0.36) MAPTEPHX2PDE2AFFAR4GPR3
SCHEMBL7772178 0.76 GRIN2B (0.33) EPHX2FFAR1FFAR4GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 67 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263749-B1 DIBENZOFURAN AND DIBENZOTHIOPHENE DERIVATIVES MERCK PATENT GMBH (DE) 2025-06-18 EP disclosed
US-20250134907-A1 FUSED DIAZEPINES AS AGONISTS OF THE INSULIN-LIKE 3 (INSL3) PEPTIDE RECEPTOR RXFP2 AND METHODS OF USE THEREOF THE UNITED STATES OF AMERICA,AS REPRESENTED BY THE SECRETARY,DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2025-05-01 US disclosed
EP-4476222-A1 FUSED DIAZEPINES AS AGONISTS OF THE INSULIN-LIKE 3 (INSL3) PEPTIDE RECEPTOR RXFP2 AND METHODS OF USE THEREOF The United States of America, as represented by the Secretary, Department of Health and Human Services (US) 2024-12-18 EP disclosed
CN-117164436-A Method for synthesizing polyfluorophenol by lanthanum cerium copper catalysis 浙江大学衢州研究院 2023-12-05 CN disclosed
CN-117024254-A Synthesis method of polyfluorophenol 浙江大学衢州研究院 2023-11-10 CN disclosed
EP-4263749-A1 DIBENZOFURAN AND DIBENZOTHIOPHENE DERIVATIVES Merck Patent GmbH (DE) 2023-10-25 EP disclosed
CN-116670255-A Dibenzofuran and dibenzothiophene derivatives 默克专利股份有限公司 2023-08-29 CN disclosed
WO-2023154197-A1 FUSED DIAZEPINES AS AGONISTS OF THE INSULIN-LIKE 3 (INSL3) PEPTIDE RECEPTOR RXFP2 AND METHODS OF USE THEREOF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2023-08-17 WO disclosed
WO-2022128847-A1 DIBENZOFURAN AND DIBENZOTHIOPHENE DERIVATIVES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed
US-11254647-B2 Benzo-fused heterocyclic derivatives useful as agonists of GPR120 JANSSEN PHARMACEUTICA NV (BE) 2022-02-22 US disclosed
US-20060025615-A1 Method for production naphthalene derivatives MERCK PATENT GMBH (DE) 2006-02-02 US disclosed
EP-1581469-A1 METHOD FOR PRODUCING NAPHTHALENE DERIVATIVES MERCK PATENT GmbH (DE) 2005-10-05 EP disclosed
US-20040173776-A1 for displays with very low threshold voltages and at the same time high values for the voltage holding ratio MERCK PATENT GMBH (DE) 2004-09-09 US disclosed
EP-1454975-A2 Liquid crystalline medium MERCK PATENT GmbH (DE) 2004-09-08 EP disclosed
WO-2004050594-A1 METHOD FOR PRODUCING NAPHTHALENE DERIVATIVES MERCK PATENT GMBH (DE) 2004-06-17 WO disclosed
US-6337034-B1 COMPOUNDS HAVING WIDE TEMPERATURE RANGE OF LIQUID CRYSTAL PHASE, LOW VISCOSITY, LOW THRESHOLD VOLTAGE AND EXCELLENT STABILITY, WHICH ARE READILY MIXED WITH VARIOUS LIQUID CRYSTAL MATERIALS AND GOOD IN SOLUBILITY AT LOW TEMPERATURE CHISSO CORPORATION (JP) 2002-01-08 US disclosed
EP-0820976-B1 FLUORINE-SUBSTITUTED LIQUID-CRYSTAL COMPOUND, LIQUID-CRYSTAL COMPOSITION AND LIQUID-CRYSTAL DISPLAY DEVICE CHISSO CORP (JP) 2001-02-21 EP disclosed
US-6051288-A LARGE DIELECTRIC ANISOTROPY, SMALL CHANGE IN THRESHOLD VOLTAGE DEPENDING ON TEMPERATURE, AND AN IMPROVED SOLUBILITY TO OTHER LIQUID CRYSTAL MATERIALS AT LOW TEMPERATURES CHISSO CORPORATION (JP) 2000-04-18 US disclosed
EP-0885875-A1 VINYLENE COMPOUNDS AND LIQUID-CRYSTAL COMPOSITION CHISSO CORPORATION (JP) 1998-12-23 EP disclosed
EP-0820976-A1 FLUORINE-SUBSTITUTED LIQUID-CRYSTAL COMPOUND, LIQUID-CRYSTAL COMPOSITION AND LIQUID-CRYSTAL DISPLAY DEVICE CHISSO CORPORATION (JP) 1998-01-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250134907-A1 FUSED DIAZEPINES AS AGONISTS OF THE INSULIN-LIKE 3 (INSL3) PEPTIDE RECEPTOR RXFP2 AND METHODS OF USE THEREOF RXFP3, RXFP4, RXFP2 TAAR1 1588/4885CA12 2330/4885CA1 2587/4885
US-20060025615-A1 Method for production naphthalene derivatives AOX1, AOC3, CBR3 TAAR1 2102/4885CA12 1271/4885CA1 1248/4885
US-11254647-B2 Benzo-fused heterocyclic derivatives useful as agonists of GPR120 GPR119, GPR180, GPR55 TAAR1 294/4885CA12 4456/4885CA1 4805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.