SCHEMBL7647137

SCHEMBL7647137

COc1ccccc1-c1csc(C(N)=O)c1S(N)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.43
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
ATP4A P20648 2/20 0.40
ATP4B P51164 2/20 0.40
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTK2 Q05397 2/20 0.38
MAP2 P11137 1/20 0.38
CDC7 O00311 1/20 0.38
HPGDS O60760 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.37
SLC9A1 P19634 1/20 0.37
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6909617 0.90 CA2 (0.41) IKBKBCA2CA9CA12CA1
SCHEMBL7643298 0.89 ALDH1A1 (0.43) IKBKBCA2CA12CA1ALDH1A1
SCHEMBL7646547 0.82 CA12 (0.42) IKBKBCA2CA9CA12CA1
SCHEMBL7640481 0.82 HTR2B (0.47) CA2CA9CA12CA1ALDH1A1
SCHEMBL7641014 0.79 CA12 (0.46) CA2CA9CA12CA1LMNA
SCHEMBL7643245 0.78 CYP3A4 (0.41) CA2CA9CA1ALDH1A1GAA
SCHEMBL28012573 0.75 BCAT2 (0.57) IKBKBATP4AATP4BALDH1A1GAA
SCHEMBL6998322 0.72 ALDH1A1 (0.46) IKBKBCA2CA9CA12CA1
SCHEMBL8187620 0.71 KDM4E (0.51) IKBKBALDH1A1GAAHPGDHSD17B10
SCHEMBL10364777 0.70 LMNA (0.62) ALDH1A1HPGDKMT2APOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6432994-B1 CARDIOVASCULAR DISORDERS, GLAUCOMA; ANTIINFLAMMATORY, WOUND HEALING, HYPOTENSIVE, ANTIASTHMATIC, AND ANTIANAPHYLACTIC AGENTS TEXAS BIOTECHNOLOGY CORPORATION 2002-08-13 US disclosed
EP-0699191-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-03-06 EP disclosed
WO-1994027979-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN IMMUNOPHARMACEUTICS, INC. (US) 1994-12-08 WO disclosed