SCHEMBL7721375

SCHEMBL7721375

CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1ccc(Br)c2ccc(O[Si](C)(C)C(C)(C)C)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
THRB P10828 1/20 0.43
CA2 P00918 1/20 0.43
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
PLIN1 O60240 1/20 0.43
RAB9A P51151 1/20 0.43
PLIN5 Q00G26 1/20 0.43
ABHD5 Q8WTS1 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
AAK1 Q2M2I8 4/20 0.40
KLK5 Q9Y337 1/20 0.40
HDAC8 Q9BY41 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL7721379 0.89 AAK1 (0.41) KDM4EALDH1A1MAPTSMN1; SMN2CTSS
SCHEMBL7718633 0.86 ALDH1A1 (0.47) KDM4EALDH1A1HPGDLMNATHRB
SCHEMBL7714829 0.81 AAK1 (0.38) AAK1HDAC8HDAC3HDAC1HDAC2
Methane SCHEMBL7718636 0.75 HDAC4 (0.46) MAPTSMN1; SMN2CTSSCTSKAAK1
SCHEMBL31347280 0.72 KMT2A (0.53) KDM4EALDH1A1HPGDLMNATHRB
SCHEMBL7719355 0.72 HDAC4 (0.46) KDM4EMAPTSMN1; SMN2CTSSCTSK
SCHEMBL7719351 0.72 HDAC4 (0.46) KDM4EMAPTSMN1; SMN2CTSSCTSK
SCHEMBL7936792 0.71 KLK5 (0.50) KDM4EALDH1A1HPGDLMNATHRB
SCHEMBL6555173 0.70 CTSS (0.52) KDM4EALDH1A1HPGDLMNATHRB
SCHEMBL6556874 0.70 CTSS (0.54) KDM4EALDH1A1HPGDLMNACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed