SCHEMBL7733852

SCHEMBL7733852

NCCC[C@@H](N)CN(C(=O)C(F)(F)F)[C@H](CCc1ccccc1)C(O)c1nc2cc(Cl)ccc2o1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
XDH P47989 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.33
CETP P11597 3/20 0.32
P2RY14 Q15391 3/20 0.32
DAGLA Q9Y4D2 1/20 0.32
HDAC1 Q13547 1/20 0.32
METAP2 P50579 1/20 0.31
AKR1B1 P15121 1/20 0.31
CASP3 P42574 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31
KIF11 P52732 2/20 0.30
MAP1LC3B Q9GZQ8 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30
KCNH2 Q12809 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7731117 0.90 FAAH (0.35) XDHDAGLAHDAC1
SCHEMBL7732045 0.89 CTSL (0.36) DAGLA
SCHEMBL7734187 0.88 F9 (0.30) METAP2
Trifluoroacetic Acid SCHEMBL7733845 0.78 LMNA (0.39) LMNAKMT2AXDHSMN1; SMN2TP53
SCHEMBL7734130 0.77 IDO1 (0.39) KMT2ADAGLAHDAC1CYP3A4CYP2C19
SCHEMBL7723163 0.76 HPGD (0.39) KMT2ASMN1; SMN2CYP2C19
SCHEMBL7732452 0.75 LMNA (0.42) LMNAKMT2AXDHSMN1; SMN2TP53
SCHEMBL7736136 0.74 XDH (0.46) LMNAKMT2AXDHSMN1; SMN2TP53
SCHEMBL7858147 0.74 XDH (0.46) LMNAKMT2AXDHSMN1; SMN2TP53
SCHEMBL7731051 0.70 LMNA (0.39) LMNAKMT2ATP53CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed