SCHEMBL7779242

SCHEMBL7779242

CC(=O)[AsH]c1ccc2[nH]c3cc(OCCNc4ccccc4CCO)ccc3c2c1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 12/20 0.38
MTNR1B P49286 11/20 0.38
KDM4E B2RXH2 2/20 0.34
MAOA P21397 1/20 0.34
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
LMNA P02545 1/20 0.33
MCL1 Q07820 1/20 0.33
DYRK1A Q13627 1/20 0.33
LTA4H P09960 1/20 0.33
PLA2G2A P14555 1/20 0.33
GPR17 Q13304 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7070543 0.85 MTNR1A (0.50) MTNR1AMTNR1BKDM4EMAOAALDH1A1
SCHEMBL6905932 0.84 CTSV (0.41) KDM4EMAOAALDH1A1HPGDMCL1
SCHEMBL7072937 0.82 KIF11 (0.36) MTNR1AMTNR1BKDM4EMAOAALDH1A1
SCHEMBL7779239 0.76 ALOX15 (0.48) KDM4EALDH1A1
SCHEMBL7781300 0.75 NR1I2 (0.33) KDM4EMAOAALDH1A1HPGDMCL1
SCHEMBL7069437 0.75 KDM4E (0.42) MTNR1AMTNR1BKDM4EMAOAALDH1A1
SCHEMBL7977146 0.72 TP53 (0.38) KDM4EALDH1A1HPGDLMNA
SCHEMBL7980657 0.72 HTR1D (0.35) MTNR1AMTNR1B
SCHEMBL7068692 0.71 ADRB2 (0.39) KDM4EALDH1A1HPGD
SCHEMBL7778752 0.71 KDM4E (0.38) KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1128845-A1 COMBINATIONS COMPRISING A BETA-AGONIST AND A FURTHER ANTDIABETIC AGENT SMITHKLINE BEECHAM PLC (GB) 2001-09-05 EP disclosed
WO-2000027434-A1 COMBINATIONS COMPRISING A BETA-AGONIST AND A FURTHER ANTIDIABETIC AGENT SMITHKLINE BEECHAM P.L.C. (GB) 2000-05-18 WO disclosed