SCHEMBL7783570

SCHEMBL7783570

Cc1oncc1OC(=O)Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.63
RAB9A P51151 3/20 0.63
HTT P42858 2/20 0.63
NPC1 O15118 2/20 0.63
GMNN O75496 1/20 0.63
LMNA P02545 1/20 0.63
TP53 P04637 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
HTR1A P08908 1/20 0.63
THRB P10828 1/20 0.63
PIM1 P11309 1/20 0.63
CYP2C9 P11712 1/20 0.63
MAOA P21397 1/20 0.63
SLC6A2 P23975 1/20 0.63
HTR2A P28223 1/20 0.63
AGTR1 P30556 1/20 0.63
CCKBR P32239 1/20 0.63
MC4R P32245 1/20 0.63
CYP2C19 P33261 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2787802 0.86 DHODH (0.48) DHODHRAB9AHTTNPC1GMNN
SCHEMBL10648551 0.84 SMN1; SMN2 (0.44) DHODHRAB9AHTTNPC1GMNN
SCHEMBL6932048 0.84 MAPT (0.46) DHODHRAB9AHTTNPC1GMNN
SCHEMBL6931877 0.83 THRB (0.48) DHODHRAB9AHTTNPC1GMNN
SCHEMBL8822110 0.82 ALDH1A1 (0.51) RAB9AHTTNPC1BLMSMN1; SMN2
SCHEMBL10646741 0.82 DHODH (0.43) DHODHRAB9AHTTNPC1GMNN
SCHEMBL10644685 0.80 NPC1 (0.41) DHODHRAB9AHTTNPC1GMNN
SCHEMBL6936296 0.80 RAB9A (0.39) DHODHRAB9AHTTNPC1GMNN
SCHEMBL6937152 0.80 CA1 (0.40) DHODHRAB9AHTTNPC1GMNN
SCHEMBL10643669 0.78 NPC1 (0.38) DHODHRAB9AHTTNPC1GMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0987256-B1 Crystal form of N-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamid AVENTIS PHARMA GMBH (DE) 2001-10-17 EP disclosed
EP-0987256-A1 Crystal form of N-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamid Hoechst Marion Roussel Deutschland GmbH (DE) 2000-03-22 EP disclosed