SCHEMBL7785656

SCHEMBL7785656

COc1ccc(C(NC(=O)c2ccc(F)cc2)c2cccc(Nc3c(N)c(=O)c3=O)c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.62
GAA P10253 2/20 0.62
LMNA P02545 3/20 0.54
SLC6A9 P48067 4/20 0.51
SLC6A5 Q9Y345 4/20 0.51
CYP3A4 P08684 2/20 0.50
KMT2A Q03164 5/20 0.45
TP53 P04637 2/20 0.45
MEN1 O00255 3/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
PKM P14618 1/20 0.42
KDM4E B2RXH2 2/20 0.40
HTT P42858 2/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
PAX8 Q06710 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7780394 0.92 ALDH1A1 (0.67) ALDH1A1GAALMNASLC6A9SLC6A5
SCHEMBL7789410 0.92 ALDH1A1 (0.57) ALDH1A1GAALMNASLC6A9SLC6A5
SCHEMBL7785458 0.90 ALDH1A1 (0.64) ALDH1A1GAALMNASLC6A9SLC6A5
SCHEMBL7784878 0.81 ALDH1A1 (0.68) ALDH1A1GAALMNASLC6A9SLC6A5
SCHEMBL7789205 0.81 GPR88 (0.48) ALDH1A1GAALMNACYP3A4KMT2A
Hydrochloric Acid SCHEMBL7785333 0.81 ALDH1A1 (0.74) ALDH1A1GAALMNASLC6A9SLC6A5
SCHEMBL7787169 0.81 ALDH1A1 (0.58) ALDH1A1GAALMNASLC6A9SLC6A5
SCHEMBL7789413 0.80 RXFP1 (0.44) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7780389 0.79 KMT2A (0.41) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7780560 0.79 ALDH1A1 (0.44) ALDH1A1GAALMNAKMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed