SCHEMBL7787169

SCHEMBL7787169

COc1ccc(C(NC(=O)c2ccccc2)c2cccc(Nc3c(OC)c(=O)c3=O)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
GAA P10253 2/20 0.58
LMNA P02545 1/20 0.58
CYP3A4 P08684 1/20 0.56
KMT2A Q03164 3/20 0.48
TP53 P04637 1/20 0.48
KCNK9 Q9NPC2 1/20 0.46
RXFP1 Q9HBX9 1/20 0.45
SLC6A9 P48067 1/20 0.45
SLC6A5 Q9Y345 1/20 0.45
ALPL P05186 1/20 0.43
GLA P06280 1/20 0.43
ALPI P09923 1/20 0.43
ALPG P10696 1/20 0.43
HSD17B2 P37059 1/20 0.43
MEN1 O00255 2/20 0.43
POLB P06746 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
NLRP3 Q96P20 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7785458 0.91 ALDH1A1 (0.64) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7784878 0.91 ALDH1A1 (0.68) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7789410 0.89 ALDH1A1 (0.57) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7785313 0.87 GPR88 (0.49) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7788988 0.86 ALDH1A1 (0.47) ALDH1A1GAALMNAKMT2AKCNK9
SCHEMBL7785061 0.82 KMT2A (0.44) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7785160 0.81 ADRB3 (0.46) ALDH1A1GAALMNAKMT2AMEN1
SCHEMBL7785656 0.81 ALDH1A1 (0.62) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7780394 0.80 ALDH1A1 (0.67) ALDH1A1GAALMNACYP3A4KMT2A
SCHEMBL7784885 0.80 KMT2A (0.43) ALDH1A1GAALMNACYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed