SCHEMBL7798890

SCHEMBL7798890

CCS(NC(=O)c1ccc(OC)cc1)(SCC(NC(=O)c1ccc(OC)cc1)C(=O)NCCc1ccccc1)C(=O)NCCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.48
RAB9A P51151 5/20 0.48
ALDH1A1 P00352 2/20 0.48
CTSS P25774 6/20 0.46
CTSK P43235 4/20 0.46
CTSL P07711 4/20 0.45
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
MAPT P10636 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
CAPN1 P07384 1/20 0.43
GAA P10253 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7793398 0.92 L3MBTL1 (0.46) NPC1RAB9AALDH1A1CTSSCTSK
SCHEMBL7798895 0.90 NPC1 (0.50) NPC1RAB9ACTSSCTSKCTSL
SCHEMBL7798884 0.83 ALDH1A1 (0.58) NPC1RAB9AALDH1A1CTSSCTSK
SCHEMBL7793442 0.80 POLB (0.43) ALDH1A1CTSSCTSKKMT2AMEN1
SCHEMBL7799269 0.80 MTNR1A (0.45) TAAR1
SCHEMBL7793458 0.77 MMP1 (0.49) ALDH1A1KMT2ASMN1; SMN2MAPTGAA
SCHEMBL7802324 0.76 ITGB3 (0.48)
SCHEMBL7803207 0.73 POLB (0.43) KMT2A
SCHEMBL7793421 0.73 POLB (0.43) KMT2A
SCHEMBL2247378 0.72 ADAMTS5 (0.59) NPC1RAB9AALDH1A1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1143960-A2 CYSTINE DERIVATIVES AS THERAPEUTIC AGENTS FOR MATRIX METALLOPROTEASE RELATED DISEASES Roche Diagnostics GmbH (DE) 2001-10-17 EP disclosed
WO-2000027378-A2 CYSTINE DERIVATIVES AS THERAPEUTIC AGENTS FOR MATRIX METALLOPROTEASE RELATED DISEASES ROCHE DIAGNOSTICS GMBH (DE) 2000-05-18 WO disclosed