SCHEMBL7828179

SCHEMBL7828179

COc1ccc(Cn2nnc(C(=O)c3ccc(NC(=O)OCc4ccccc4)cc3)c2C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 9/20 0.53
PTGDR2 Q9Y5Y4 3/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 2/20 0.47
PTGER4 P35408 1/20 0.46
HTT P42858 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
POLB P06746 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7824962 0.92 AKR1C3 (0.51) AKR1C3PTGDR2MEN1KMT2AALDH1A1
SCHEMBL7828177 0.86 AKR1C3 (0.47) AKR1C3MEN1KMT2AALDH1A1PTGER4
SCHEMBL7829631 0.84 AKR1C3 (0.51) AKR1C3MEN1KMT2AALDH1A1PTGER4
SCHEMBL7824961 0.80 CYP19A1 (0.46) AKR1C3ALDH1A1ADORA3NPC1RAB9A
SCHEMBL1223807 0.77 RAB9A (0.67) ALDH1A1HTTNPC1RAB9APOLB
SCHEMBL8073566 0.76 CASP3 (0.44) AKR1C3MEN1KMT2AHTT
SCHEMBL7822920 0.76 AKR1C3 (0.42) AKR1C3KMT2AALDH1A1PTGER4HTT
SCHEMBL7829626 0.74 AKR1C3 (0.49) AKR1C3MEN1KMT2AALDH1A1PTGER4
SCHEMBL11813314 0.74 TP53 (0.68) ALDH1A1HTTNPC1RAB9APOLB
SCHEMBL7816139 0.74 ALOX15 (0.51) AKR1C3MEN1KMT2AALDH1A1PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686636-B1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA CO (JP) 2001-04-04 EP disclosed
US-5840895-A INTERMEDIATES FOR ANTIALLERGENS MEIJI SEIKA KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
EP-0686636-A1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA KABUSHIKI KAISHA (JP) 1995-12-13 EP disclosed