SCHEMBL7834854

SCHEMBL7834854

COc1ccc(Br)cc1CC(NC(=O)CNC(=O)c1cccc(NC=NN)c1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR139 Q6DWJ6 3/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 2/20 0.41
MAPT P10636 3/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
ITGB3 P05106 2/20 0.40
ITGAV P06756 2/20 0.40
ITGB1 P05556 1/20 0.40
ITGA2B P08514 1/20 0.40
ITGB5 P18084 1/20 0.40
PPARG P37231 2/20 0.39
PPARD Q03181 2/20 0.39
PPARA Q07869 2/20 0.39
LMNA P02545 2/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7823384 0.91 ALDH1A1 (0.40) GPR139SMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL7345869 0.88 HTT (0.43) GPR139SMN1; SMN2KDM4EMAPTNPC1
SCHEMBL7339213 0.86 MEN1 (0.46) KDM4EMAPTNPC1GAARAB9A
SCHEMBL6773894 0.85 ITGB3 (0.47) GPR139KDM4EITGB3ITGAVITGB1
SCHEMBL6779571 0.84 FPR2 (0.43) NPC1GAARAB9AITGB3ITGAV
SCHEMBL7347036 0.84 HPGD (0.42) GPR139SMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL6773776 0.83 CTSB (0.43) KDM4EMAPTNPC1GAARAB9A
SCHEMBL6778010 0.82 GPR139 (0.49) GPR139SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL6782093 0.81 ITGB1 (0.41) GPR139ITGB3ITGAVITGB1ITGB5
SCHEMBL7340359 0.81 GPR139 (0.40) GPR139SMN1; SMN2MAPTITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP claimed