SCHEMBL7862023

SCHEMBL7862023

N=C(N)Nc1ccc(S(=O)(=O)CNc2cccc(C(CC(=O)O)c3ccccc3)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 7/20 0.39
ITGB3 P05106 2/20 0.39
ITGA2B P08514 2/20 0.39
SCN3A Q9NY46 1/20 0.38
CA12 O43570 6/20 0.37
CA1 P00915 6/20 0.37
CA9 Q16790 6/20 0.37
HPN P05981 2/20 0.37
HTT P42858 2/20 0.37
PLAU P00749 1/20 0.37
CA4 P22748 2/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862026 0.83 CA2 (0.36) CA2ITGB3SCN3ACA12CA1
SCHEMBL7862046 0.79 ITGB3 (0.45) CA2ITGB3CA1POLBMAPT
SCHEMBL7862025 0.78 TSHR (0.52) HTTPOLBMAPTALDH1A1LMNA
SCHEMBL7863273 0.78 FFAR1 (0.43) ITGB3ITGA2BPOLBMAPTLMNA
SCHEMBL7856539 0.77 ITGB3 (0.41) CA2ITGB3CA12CA1CA9
SCHEMBL7856433 0.76 ITGB3 (0.54) ITGB3ITGA2BHTTPLAUPOLB
SCHEMBL7455765 0.75 ITGB3 (0.58) ITGB3ITGA2BPLAUPOLBALDH1A1
SCHEMBL7863285 0.74 ITGB3 (0.48) ITGB3ITGA2BPOLBMAPTALDH1A1
SCHEMBL7861944 0.73 HDAC1 (0.45) ITGB3ITGA2BPOLBMAPTALDH1A1
SCHEMBL7856431 0.73 HDAC1 (0.45) ITGB3ITGA2BPOLBMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed