SCHEMBL7862025

SCHEMBL7862025

CN(c1cccc(C(CC(=O)O)c2ccccc2)c1)S(=O)(=O)c1ccc(NC(=N)N)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
MAPT P10636 9/20 0.50
KMT2A Q03164 8/20 0.50
MEN1 O00255 7/20 0.50
LMNA P02545 6/20 0.50
HTT P42858 4/20 0.50
SMN1; SMN2 Q16637 4/20 0.50
POLB P06746 2/20 0.47
ALOX12 P18054 3/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 8/20 0.45
GPR27 Q9NS67 1/20 0.45
ABCC9 O60706 1/20 0.45
ABCC8 Q09428 1/20 0.45
KCNJ11 Q14654 1/20 0.45
KCNJ8 Q15842 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MAPK1 P28482 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862023 0.78 CA2 (0.39) MAPTLMNAHTTPOLBALDH1A1
SCHEMBL7856539 0.74 ITGB3 (0.41) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL7862046 0.74 ITGB3 (0.45) MAPTKMT2AMEN1POLB
SCHEMBL8534762 0.72 MMP1 (0.39) TSHRMAPTKMT2AMEN1LMNA
SCHEMBL7455765 0.72 ITGB3 (0.58) KMT2AMEN1POLBALDH1A1
SCHEMBL9408034 0.71 TSHR (0.72) TSHRMAPTKMT2AMEN1LMNA
SCHEMBL7863285 0.71 ITGB3 (0.48) MAPTLMNAPOLBALDH1A1MAPK1
SCHEMBL12010879 0.71 TSHR (0.81) TSHRMAPTKMT2AMEN1LMNA
SCHEMBL7856431 0.70 HDAC1 (0.45) MAPTKMT2AMEN1LMNASMN1; SMN2
SCHEMBL7856433 0.70 ITGB3 (0.54) MAPTKMT2AMEN1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed