SCHEMBL7910125

SCHEMBL7910125

BCC1=CN2C=C(C)NC2C(c2cccc(Cl)c2)=C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 5/20 0.34
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33
TP53 P04637 2/20 0.32
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
ESR2 Q92731 1/20 0.31
MAPT P10636 2/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
DRD2 P14416 1/20 0.30
DRD4 P21917 1/20 0.30
DRD3 P35462 1/20 0.30
IKBKE Q14164 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7930844 0.80 PGR (0.33) PGRALDH1A1POLBAPOBEC3GTP53
SCHEMBL7913037 0.80 SLC6A3 (0.35) PGRALDH1A1MEN1KMT2AMAPT
SCHEMBL7902988 0.78 GRIN1 (0.32) NPC1RAB9ACYP1A2CYP2C9CYP2C19
SCHEMBL7915334 0.78 DHFR (0.32) NPC1RAB9ASMN1; SMN2IKBKE
SCHEMBL7902852 0.76 NPC1 (0.34) POLBTP53KMT2ANPC1RAB9A
SCHEMBL7902845 0.76 PIM1 (0.31)
SCHEMBL7912990 0.74 PARP1 (0.37) ALDH1A1MEN1KMT2AMAPTHTT
SCHEMBL7913078 0.72 DYRK3 (0.37)
SCHEMBL7917981 0.71 DYRK3 (0.35) ALDH1A1POLBMEN1KMT2ARAB9A
SCHEMBL7916997 0.71 JAK2 (0.35) ALDH1A1TP53KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed