SCHEMBL7920535

SCHEMBL7920535

CC1=C(C)N2C=C(Cc3ccc(N)nc3)C=C(c3cccc(Cl)c3)C2N1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.33
PTPN11 Q06124 1/20 0.32
IKBKE Q14164 1/20 0.31
STK4 Q13043 1/20 0.31
STK3 Q13188 1/20 0.31
LRRK2 Q5S007 1/20 0.31
HRH1 P35367 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913175 0.88 MAOB (0.33) IKBKESTK4STK3LRRK2TAAR1
SCHEMBL7915334 0.84 DHFR (0.32) DHFRPTPN11IKBKESTK4STK3
SCHEMBL7911726 0.82
SCHEMBL7915330 0.81 MEN1 (0.36)
SCHEMBL7902850 0.79 PGR (0.33)
SCHEMBL7902988 0.73 GRIN1 (0.32)
SCHEMBL7917010 0.72 MAOB (0.33) IKBKESTK4STK3LRRK2TAAR1
SCHEMBL7911301 0.72 NLRP3 (0.35)
SCHEMBL7911681 0.72 MAPT (0.36)
SCHEMBL7902852 0.71 NPC1 (0.34) STK4STK3LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed