SCHEMBL7932225

SCHEMBL7932225

COc1cc(CNC(=O)CS)ccc1O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.66
CYP3A4 P08684 3/20 0.66
CYP2D6 P10635 2/20 0.66
CYP2C9 P11712 2/20 0.66
CYP2C19 P33261 2/20 0.66
BLM P54132 2/20 0.66
PMP22 Q01453 2/20 0.66
ALDH1A1 P00352 2/20 0.66
ALOX15 P16050 2/20 0.66
HPGD P15428 1/20 0.66
TRPV1 Q8NER1 6/20 0.65
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
POLB P06746 1/20 0.62
TSHR P16473 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
KDM1A O60341 1/20 0.58
NR1I2 O75469 1/20 0.58
LMNA P02545 1/20 0.58
ALOX5 P09917 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8168115 0.87 ALDH1A1 (0.67) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL17205705 0.87 CYP1A2 (0.71) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL24092698 0.85 CYP1A2 (0.66) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5348698 0.84 CYP1A2 (0.90) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL906527 0.84 CYP1A2 (0.81) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5707095 0.83 MTNR1A (0.69) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL297477 0.83 ALDH1A1 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7528872 0.83 ERCC1 (0.73) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL18517554 0.83 CYP1A2 (0.70) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7529264 0.83 ERCC1 (0.73) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110190285-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT ABSOLUTE SCIENCE, INC. (US) 2011-08-04 US disclosed
US-20110034521-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-02-10 US disclosed
WO-2010033360-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT 1/3 ABSOLUTE SCIENCE, INC. (US) 2010-03-25 WO disclosed
WO-2009045761-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES ABSOLUTE SCIENCE, INC. (US) 2009-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034521-A1 COMPOUNDS AND METHODS FOR TREATING ZINC MATRIX METALLOPROTEASE DEPENDENT DISEASES MMP7, MMP3, MMP9 CYP1A2 1547/4885CYP3A4 3370/4885CYP2D6 2162/4885
US-20110190285-A1 METHODS OF TREATING A BOTULINUM TOXIN RELATED CONDITION IN A SUBJECT NPY5R, RAC3, CPA3 CYP1A2 927/4885CYP3A4 2145/4885CYP2D6 1496/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.