SCHEMBL7933428

SCHEMBL7933428

CCC[C@@](C)(C(=O)NNCC(C)C)[C@H](CC=Cc1ccccc1)C(=O)NOC1CCCCO1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.33
CTSC P53634 1/20 0.33
TGFBR1 P36897 1/20 0.32
MGLL Q99685 1/20 0.32
SLC6A3 Q01959 2/20 0.31
LNPEP Q9UIQ6 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6944688 0.83 P2RX3 (0.31) P2RX3CTSCTGFBR1CCNA2CDK2
SCHEMBL7933480 0.80 KDM4E (0.33) TGFBR1SLC6A3
SCHEMBL6983937 0.80 ADAM17 (0.42) P2RX3CTSCTGFBR1MGLLSLC6A3
SCHEMBL6984895 0.78 CTSC (0.33) P2RX3CTSCTGFBR1MGLL
SCHEMBL6948116 0.76 TGFBR1 (0.32) P2RX3CTSCTGFBR1MGLL
SCHEMBL7930228 0.75 CTSC (0.33) P2RX3CTSCTGFBR1MGLLSLC6A3
SCHEMBL6941960 0.75 ADAM17 (0.33) P2RX3CTSCTGFBR1MGLLCCNA2
SCHEMBL7937958 0.75 P2RX3 (0.31) P2RX3TGFBR1
SCHEMBL7928806 0.75 P2RX3 (0.34) P2RX3CTSCTGFBR1MGLLSLC6A3
SCHEMBL7940268 0.75 P2RX3 (0.30) P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed