SCHEMBL7953114

SCHEMBL7953114

CCc1ccc(OCCC(O)N2CCC(c3cccnc3)CC2)cc1.O=S(=O)(O)c1cccc2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 3/20 0.35
P2RX7 Q99572 7/20 0.34
ROCK2 O75116 3/20 0.34
ROCK1 Q13464 3/20 0.34
TP53 P04637 1/20 0.34
KMT2A Q03164 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7953116 0.85 MAPT (0.47) ADRB3KMT2A
SCHEMBL7953119 0.75 HTR7 (0.40) P2RX7
SCHEMBL7965925 0.67 HTR1A (0.47)
SCHEMBL7953252 0.64 CCR2 (0.35)
Fumaric Acid SCHEMBL7967350 0.62 RAB9A (0.42) KMT2A
SCHEMBL7966382 0.62 OPRL1 (0.43) KMT2A
SCHEMBL16218244 0.60 CYP11B2 (0.57)
Pyridine SCHEMBL1270547 0.59 CA1 (0.50) KMT2A
Pyridine SCHEMBL1270544 0.59 CA1 (0.50) KMT2A
Alcohol SCHEMBL282185 0.59 CA1 (0.53) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
WO-2000006166-A1 5-HT1F ANTAGONISTS ELI LILLY AND COMPANY (US) 2000-02-10 WO disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed