SCHEMBL7953266

SCHEMBL7953266

Cc1ccc(OC(O)CCN2CCC(OC(=O)CC(=O)OC3(c4cncc5ccccc45)CCN(CCC(O)Oc4ccc(C)c(C)c4)CC3)(c3cncc4ccccc34)CC2)cc1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.34
DRD3 P35462 3/20 0.34
DRD2 P14416 2/20 0.34
CYP11B2 P19099 2/20 0.34
CYP11B1 P15538 1/20 0.33
OPRM1 P35372 2/20 0.32
OPRL1 P41146 2/20 0.32
OPRD1 P41143 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
HTR7 P34969 2/20 0.32
HTR1A P08908 1/20 0.32
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MMP1 P03956 1/20 0.31
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
FAAH O00519 1/20 0.31
POLB P06746 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963764 0.79 MEN1 (0.35) CCR5DRD3CYP11B2ITGA4ITGB7
SCHEMBL7965454 0.78 OPRL1 (0.36) DRD3OPRM1OPRL1HTR1A
SCHEMBL7965779 0.78 ITGA4 (0.33) CCR5DRD3DRD2CYP11B2CYP11B1
SCHEMBL8139378 0.75 SLC6A1 (0.34) CCR5DRD3DRD2CYP11B2OPRM1
SCHEMBL7963100 0.75 SLC6A1 (0.34) CCR5DRD3DRD2CYP11B2OPRM1
SCHEMBL7967096 0.74 TUBB4A (0.38) CYP11B2CYP11B1OPRM1OPRL1OPRD1
SCHEMBL7962999 0.71 OPRL1 (0.40) DRD2OPRM1OPRL1OPRD1HTR1A
SCHEMBL7969481 0.71 LTA4H (0.38) DRD3DRD2OPRM1OPRL1OPRD1
SCHEMBL7965995 0.71
Malonic Acid SCHEMBL7953260 0.70 MAPT (0.44) HTR1ALMNASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed