SCHEMBL7963764

SCHEMBL7963764

C=CC(=O)OC1(c2cncc3ccccc23)CCN(CCC(O)Oc2ccc(OC)cc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CCR5 P51681 2/20 0.34
HTR1A P08908 3/20 0.33
SLC6A1 P30531 1/20 0.33
SLC6A12 P48065 1/20 0.33
SLC6A11 P48066 1/20 0.33
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
HTT P42858 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2B P41595 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
DRD3 P35462 1/20 0.32
CYP11B2 P19099 1/20 0.32
TUBB4A P04350 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963760 0.84 KDM4E (0.45) MEN1KMT2AHTR1AHTT
SCHEMBL7953266 0.79 CCR5 (0.34) CCR5HTR1AITGA4ITGB7HTR2A
SCHEMBL7963100 0.76 SLC6A1 (0.34) MEN1KMT2ACCR5HTR1ASLC6A1
SCHEMBL8139378 0.76 SLC6A1 (0.34) MEN1KMT2ACCR5HTR1ASLC6A1
SCHEMBL7965454 0.75 OPRL1 (0.36) MEN1KMT2AHTR1ASLC6A1SLC6A12
SCHEMBL7965779 0.74 ITGA4 (0.33) CCR5HTR1AITGA4ITGB7ADRA1A
SCHEMBL7962999 0.72 OPRL1 (0.40) HTR1A
SCHEMBL7967096 0.72 TUBB4A (0.38) SLC6A1SLC6A12SLC6A11ADRA1AADRA1B
Acrylic Acid SCHEMBL7963757 0.69 ALDH1A1 (0.38) MEN1KMT2AITGA4ITGB7HTT
SCHEMBL7966082 0.68 KDM4E (0.48) MEN1KMT2AHTR1AHTR2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed