SCHEMBL7990102

SCHEMBL7990102

COc1c(C(=O)Nc2cccc3c2CCN(C)C3C)cccc1C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.46
HTR1F P30939 1/20 0.38
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 3/20 0.38
NPSR1 Q6W5P4 3/20 0.38
TSHR P16473 3/20 0.38
HSD17B10 Q99714 2/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 3/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
GAA P10253 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993333 0.80 NR1H4 (0.45) NR1H4KDM4EALDH1A1NPSR1POLB
SCHEMBL7979061 0.76 PDE4D (0.39) KDM4EALDH1A1POLBRAB9ASMN1; SMN2
SCHEMBL7993247 0.76 KDM4E (0.43) KDM4EALDH1A1NPSR1TSHRHSD17B10
SCHEMBL8012751 0.75 ADRA2A (0.46) ALDH1A1POLBHPGDNPC1RAB9A
SCHEMBL8025490 0.73 DRD2 (0.51) KDM4EALDH1A1TSHRHSD17B10HPGD
SCHEMBL7991365 0.72 BRPF1 (0.43) KDM4EALDH1A1NPSR1POLBNPC1
SCHEMBL7993464 0.72 KMT2A (0.42) KDM4EALDH1A1NPSR1TSHRHSD17B10
SCHEMBL8025533 0.69 DRD2 (0.43)
SCHEMBL22863188 0.69 DRD1 (0.41) KMT2AMEN1
SCHEMBL24252069 0.69 NR1H4 (0.59) NR1H4KDM4EALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6277861-B1 FOR TREATMENT AND PROPHYLAXIS OF NERVOUS SYSTEM DISORDERS, PSYCHOLOGICAL DISORDERS, MUSCULAR DISORDERS, DRUG ADDICTION WITHDRAWAL, PAIN SMITHKLINE BEECHAM, P.L.C. (GB) 2001-08-21 US disclosed