SCHEMBL7994097

SCHEMBL7994097

O=C(Nc1[c]cccc1-c1ccccc1)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.48
HDAC7 Q8WUI4 5/20 0.48
HDAC8 Q9BY41 5/20 0.48
HDAC6 Q9UBN7 5/20 0.48
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
TACR1 P25103 1/20 0.40
ACHE P22303 1/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19065135 0.80 BCAT2 (0.44) MEN1RAB9AKMT2AALDH1A1CHRNB2
SCHEMBL10599404 0.80 HSP90AA1 (0.46) HDAC1MEN1NPC1RAB9AKMT2A
SCHEMBL7392337 0.73 SIGMAR1 (0.40) RAB9AHSD17B10ALDH1A1CHRNB2CHRNB4
SCHEMBL10969933 0.73 ALDH1A1 (0.44) MEN1TP53RAB9AKMT2AHSD17B10
SCHEMBL16936095 0.71 CHRNB2 (0.49) TP53KMT2AALDH1A1CHRNB2CHRNB4
SCHEMBL610542 0.70 L3MBTL1 (0.45) HDAC1HDAC7HDAC8HDAC6MEN1
SCHEMBL8187332 0.70 TDO2 (0.38) HDAC8HDAC6MEN1RAB9AKMT2A
SCHEMBL4056504 0.69 ALDH1A1 (0.41) HDAC8HDAC6MEN1KMT2AHSD17B10
SCHEMBL8755361 0.68 RAB9A (0.71) HDAC1HDAC7HDAC8HDAC6MEN1
SCHEMBL474941 0.67 HDAC1 (0.65) HDAC1HDAC7HDAC8HDAC6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087852-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL URACILS USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-11-22 WO claimed