SCHEMBL7995048

SCHEMBL7995048

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2N(C(=O)CN)CC21C

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.43
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.40
CYP51A1 Q16850 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
CCKBR P32239 3/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HPGD P15428 1/20 0.38
PYGL P06737 1/20 0.37
AKR1C3 P42330 1/20 0.37
STAT6 P42226 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8004923 0.82 PYGL (0.37) DRD2CYP51A1PYGL
SCHEMBL7998609 0.81 DRD2 (0.47) DRD2KDM4EGAACYP51A1ALDH1A1
SCHEMBL7989861 0.81 DRD2 (0.47) DRD2KDM4EGAACYP51A1ALDH1A1
SCHEMBL7995568 0.80 DRD2 (0.34) DRD2CYP51A1ALDH1A1CCKBRPYGL
SCHEMBL8002722 0.79 STAT6 (0.35) DRD2CYP51A1ALDH1A1CCKBRPYGL
SCHEMBL7989864 0.78 PYGL (0.37) DRD2CYP51A1PYGL
SCHEMBL8002404 0.78 PYGL (0.37) DRD2KDM4ECYP51A1ALDH1A1PYGL
SCHEMBL8004750 0.77 MMP2 (0.33) DRD2GAACYP51A1TAS1R3TAS1R1
SCHEMBL8004714 0.76 ALOX15 (0.40) CYP51A1PYGL
SCHEMBL8002402 0.76 STAT6 (0.37) CYP51A1ALDH1A1CCKBRPYGLSTAT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111680-A1 TRPV4 ANTAGONISTS SMITHLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed